Search

Brian E. Mcdowell

Examiner (ID: 2181, Phone: (571)270-5755 , Office: P/1624 )

Most Active Art Unit
1624
Art Unit(s)
4161, 1624
Total Applications
1622
Issued Applications
1025
Pending Applications
135
Abandoned Applications
522

Applications

Application numberTitle of the applicationFiling DateStatus
Array ( [id] => 19246908 [patent_doc_number] => 20240197892 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-06-20 [patent_title] => Chemically Coupled Transporter for Low-Hydrophobicity Bioactive Drugs into the Central Nervous System [patent_app_type] => utility [patent_app_number] => 18/590749 [patent_app_country] => US [patent_app_date] => 2024-02-28 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 14622 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -11 [patent_words_short_claim] => 41 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18590749 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/590749
Chemically Coupled Transporter for Low-Hydrophobicity Bioactive Drugs into the Central Nervous System Feb 27, 2024 Pending
Array ( [id] => 19299934 [patent_doc_number] => 20240228503 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-07-11 [patent_title] => TRIAZOLE-SUBSTITUTED IMIDAZO[1,2-A]PYRIMIDINES AS CGAS INHIBITORS [patent_app_type] => utility [patent_app_number] => 18/586620 [patent_app_country] => US [patent_app_date] => 2024-02-26 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 31156 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -27 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18586620 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/586620
Triazole-substituted imidazo[1,2-a]pyrimidines as cGAS inhibitors Feb 25, 2024 Issued
Array ( [id] => 19784138 [patent_doc_number] => 20250057817 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2025-02-20 [patent_title] => KRAS G12C INHIBITORS AND METHODS OF USING THE SAME [patent_app_type] => utility [patent_app_number] => 18/443925 [patent_app_country] => US [patent_app_date] => 2024-02-16 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 56204 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => 0 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18443925 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/443925
KRAS G12C INHIBITORS AND METHODS OF USING THE SAME Feb 15, 2024 Abandoned
Array ( [id] => 19233635 [patent_doc_number] => 20240190827 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-06-13 [patent_title] => Inhibitors of Rho Associated Coiled-Coil Containing Protein Kinase [patent_app_type] => utility [patent_app_number] => 18/434994 [patent_app_country] => US [patent_app_date] => 2024-02-07 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 22178 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -14 [patent_words_short_claim] => 367 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18434994 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/434994
Inhibitors of Rho Associated Coiled-Coil Containing Protein Kinase Feb 6, 2024 Pending
Array ( [id] => 19180997 [patent_doc_number] => 11987578 [patent_country] => US [patent_kind] => B1 [patent_issue_date] => 2024-05-21 [patent_title] => 7-(4-((5-(2-chlorobenzylideneamino)-2-thioxo-1,3,4-thiadiazol-3(2H)-yl)methyl)piperazin-1-yl)-1-cyclopropyl-6-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxylic acid as an anti-inflammatory compound [patent_app_type] => utility [patent_app_number] => 18/434601 [patent_app_country] => US [patent_app_date] => 2024-02-06 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 2 [patent_figures_cnt] => 2 [patent_no_of_words] => 3874 [patent_no_of_claims] => 1 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 24 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18434601 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/434601
7-(4-((5-(2-chlorobenzylideneamino)-2-thioxo-1,3,4-thiadiazol-3(2H)-yl)methyl)piperazin-1-yl)-1-cyclopropyl-6-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxylic acid as an anti-inflammatory compound Feb 5, 2024 Issued
Array ( [id] => 19667464 [patent_doc_number] => 12180191 [patent_country] => US [patent_kind] => B1 [patent_issue_date] => 2024-12-31 [patent_title] => 2-[(1H-benzimidazol-2-yl)imino]-5,5-diphenylimidazolidin-4-one as an antimicrobial compound [patent_app_type] => utility [patent_app_number] => 18/430400 [patent_app_country] => US [patent_app_date] => 2024-02-01 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 2 [patent_figures_cnt] => 2 [patent_no_of_words] => 3995 [patent_no_of_claims] => 1 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 113 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18430400 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/430400
2-[(1H-benzimidazol-2-yl)imino]-5,5-diphenylimidazolidin-4-one as an antimicrobial compound Jan 31, 2024 Issued
Array ( [id] => 19299896 [patent_doc_number] => 20240228465 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-07-11 [patent_title] => SUBSTITUTED PYRIDINE N-OXIDE DERIVATIVES USEFUL AS A FACTOR XIA INHIBITORS [patent_app_type] => utility [patent_app_number] => 18/428046 [patent_app_country] => US [patent_app_date] => 2024-01-31 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 32083 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -14 [patent_words_short_claim] => 462 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18428046 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/428046
SUBSTITUTED PYRIDINE N-OXIDE DERIVATIVES USEFUL AS A FACTOR XIA INHIBITORS Jan 30, 2024 Abandoned
Array ( [id] => 19642866 [patent_doc_number] => 20240417386 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-12-19 [patent_title] => INHIBITORS OF RET [patent_app_type] => utility [patent_app_number] => 18/422258 [patent_app_country] => US [patent_app_date] => 2024-01-25 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 17988 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -32 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18422258 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/422258
INHIBITORS OF RET Jan 24, 2024 Pending
Array ( [id] => 19281464 [patent_doc_number] => 20240217938 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-07-04 [patent_title] => MORPHIC FORMS OF HEXADECYLOXYPROPYL-PHOSPHONATE ESTERS AND METHODS OF SYNTHESIS THEREOF [patent_app_type] => utility [patent_app_number] => 18/414198 [patent_app_country] => US [patent_app_date] => 2024-01-16 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 32700 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -18 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18414198 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/414198
MORPHIC FORMS OF HEXADECYLOXYPROPYL-PHOSPHONATE ESTERS AND METHODS OF SYNTHESIS THEREOF Jan 15, 2024 Pending
Array ( [id] => 19571766 [patent_doc_number] => 20240376058 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-11-14 [patent_title] => GCN2 AND PERK KINASE INHIBITORS AND METHODS OF USE THEREOF [patent_app_type] => utility [patent_app_number] => 18/408956 [patent_app_country] => US [patent_app_date] => 2024-01-10 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 63809 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -26 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18408956 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/408956
GCN2 AND PERK KINASE INHIBITORS AND METHODS OF USE THEREOF Jan 9, 2024 Pending
Array ( [id] => 19112675 [patent_doc_number] => 20240124425 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-04-18 [patent_title] => SOLID STATE FORMS OF BELUMOSUDIL AND BELUMOSUDIL SALTS [patent_app_type] => utility [patent_app_number] => 18/393915 [patent_app_country] => US [patent_app_date] => 2023-12-22 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 16944 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -15 [patent_words_short_claim] => 123 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18393915 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/393915
Solid state forms of Belumosudil and Belumosudil salts Dec 21, 2023 Issued
Array ( [id] => 19403566 [patent_doc_number] => 20240287077 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-08-29 [patent_title] => PYRAZOLOPYRIMIDINE COMPOUNDS [patent_app_type] => utility [patent_app_number] => 18/391047 [patent_app_country] => US [patent_app_date] => 2023-12-20 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 12996 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -8 [patent_words_short_claim] => 65 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18391047 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/391047
PYRAZOLOPYRIMIDINE COMPOUNDS Dec 19, 2023 Abandoned
Array ( [id] => 19165789 [patent_doc_number] => 11981675 [patent_country] => US [patent_kind] => B1 [patent_issue_date] => 2024-05-14 [patent_title] => Pyrrolo[3,2-C]quinoline-2,3-dione compounds as CK2 inhibitors [patent_app_type] => utility [patent_app_number] => 18/536912 [patent_app_country] => US [patent_app_date] => 2023-12-12 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 9462 [patent_no_of_claims] => 17 [patent_no_of_ind_claims] => 3 [patent_words_short_claim] => 66 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18536912 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/536912
Pyrrolo[3,2-C]quinoline-2,3-dione compounds as CK2 inhibitors Dec 11, 2023 Issued
Array ( [id] => 19105770 [patent_doc_number] => 11958851 [patent_country] => US [patent_kind] => B1 [patent_issue_date] => 2024-04-16 [patent_title] => Pyrrolo[3,2-c]quinoline compounds as CK2 inhibitors [patent_app_type] => utility [patent_app_number] => 18/533067 [patent_app_country] => US [patent_app_date] => 2023-12-07 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 9694 [patent_no_of_claims] => 10 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 391 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18533067 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/533067
Pyrrolo[3,2-c]quinoline compounds as CK2 inhibitors Dec 6, 2023 Issued
Array ( [id] => 19135566 [patent_doc_number] => 11970496 [patent_country] => US [patent_kind] => B1 [patent_issue_date] => 2024-04-30 [patent_title] => Pyrrolo[3,2-c]quinoline compounds as CK2 inhibitors [patent_app_type] => utility [patent_app_number] => 18/533073 [patent_app_country] => US [patent_app_date] => 2023-12-07 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 9698 [patent_no_of_claims] => 11 [patent_no_of_ind_claims] => 3 [patent_words_short_claim] => 101 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18533073 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/533073
Pyrrolo[3,2-c]quinoline compounds as CK2 inhibitors Dec 6, 2023 Issued
Array ( [id] => 19157605 [patent_doc_number] => 20240150312 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-05-09 [patent_title] => PYRAZINE COMPOUND [patent_app_type] => utility [patent_app_number] => 18/532293 [patent_app_country] => US [patent_app_date] => 2023-12-07 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 51784 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => 0 [patent_words_short_claim] => 221 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18532293 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/532293
PYRAZINE COMPOUND Dec 6, 2023 Abandoned
Array ( [id] => 19543059 [patent_doc_number] => 20240360095 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-10-31 [patent_title] => NOVEL KINASE MODULATORS [patent_app_type] => utility [patent_app_number] => 18/508085 [patent_app_country] => US [patent_app_date] => 2023-11-13 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 75212 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -23 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18508085 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/508085
NOVEL KINASE MODULATORS Nov 12, 2023 Pending
18/388734 5-(SUBSTITUTEDPHENYL)-7-THIOXO-7,8-DIHYDROPYRIMIDO[4,5- d]PYRIMIDINE-2,4(1H,3H)-DIONE ANALOGUES AS ANTIBACTERIAL AGENTS Nov 9, 2023
Array ( [id] => 19135542 [patent_doc_number] => 11970472 [patent_country] => US [patent_kind] => B1 [patent_issue_date] => 2024-04-30 [patent_title] => 5-((2-isopropyl-5-methylphenoxy)methyl)-3-(naphthalen-1-yl)-1,2,4-oxadiazole as an anti-cancer and antimicrobial compound [patent_app_type] => utility [patent_app_number] => 18/386545 [patent_app_country] => US [patent_app_date] => 2023-11-02 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 4475 [patent_no_of_claims] => 10 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 8 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18386545 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/386545
5-((2-isopropyl-5-methylphenoxy)methyl)-3-(naphthalen-1-yl)-1,2,4-oxadiazole as an anti-cancer and antimicrobial compound Nov 1, 2023 Issued
Array ( [id] => 20414117 [patent_doc_number] => 12497387 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2025-12-16 [patent_title] => Process for the preparation of pyrimidinyl-4-aminopyrazole compounds [patent_app_type] => utility [patent_app_number] => 18/384080 [patent_app_country] => US [patent_app_date] => 2023-10-26 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 1730 [patent_no_of_claims] => 5 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 247 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18384080 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/384080
Process for the preparation of pyrimidinyl-4-aminopyrazole compounds Oct 25, 2023 Issued
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