
Brian E. Mcdowell
Examiner (ID: 2181, Phone: (571)270-5755 , Office: P/1624 )
| Most Active Art Unit | 1624 |
| Art Unit(s) | 4161, 1624 |
| Total Applications | 1622 |
| Issued Applications | 1025 |
| Pending Applications | 135 |
| Abandoned Applications | 522 |
Applications
| Application number | Title of the application | Filing Date | Status |
|---|---|---|---|
Array
(
[id] => 19246908
[patent_doc_number] => 20240197892
[patent_country] => US
[patent_kind] => A1
[patent_issue_date] => 2024-06-20
[patent_title] => Chemically Coupled Transporter for Low-Hydrophobicity Bioactive Drugs into the Central Nervous System
[patent_app_type] => utility
[patent_app_number] => 18/590749
[patent_app_country] => US
[patent_app_date] => 2024-02-28
[patent_effective_date] => 0000-00-00
[patent_drawing_sheets_cnt] => 0
[patent_figures_cnt] => 0
[patent_no_of_words] => 14622
[patent_no_of_claims] => 0
[patent_no_of_ind_claims] => -11
[patent_words_short_claim] => 41
[patent_maintenance] => 1
[patent_no_of_assignments] => 0
[patent_current_assignee] =>[type] => publication
[pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18590749
[rel_patent_id] =>[rel_patent_doc_number] =>) 18/590749 | Chemically Coupled Transporter for Low-Hydrophobicity Bioactive Drugs into the Central Nervous System | Feb 27, 2024 | Pending |
Array
(
[id] => 19299934
[patent_doc_number] => 20240228503
[patent_country] => US
[patent_kind] => A1
[patent_issue_date] => 2024-07-11
[patent_title] => TRIAZOLE-SUBSTITUTED IMIDAZO[1,2-A]PYRIMIDINES AS CGAS INHIBITORS
[patent_app_type] => utility
[patent_app_number] => 18/586620
[patent_app_country] => US
[patent_app_date] => 2024-02-26
[patent_effective_date] => 0000-00-00
[patent_drawing_sheets_cnt] => 0
[patent_figures_cnt] => 0
[patent_no_of_words] => 31156
[patent_no_of_claims] => 0
[patent_no_of_ind_claims] => -27
[patent_words_short_claim] => 2
[patent_maintenance] => 1
[patent_no_of_assignments] => 0
[patent_current_assignee] =>[type] => publication
[pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18586620
[rel_patent_id] =>[rel_patent_doc_number] =>) 18/586620 | Triazole-substituted imidazo[1,2-a]pyrimidines as cGAS inhibitors | Feb 25, 2024 | Issued |
Array
(
[id] => 19784138
[patent_doc_number] => 20250057817
[patent_country] => US
[patent_kind] => A1
[patent_issue_date] => 2025-02-20
[patent_title] => KRAS G12C INHIBITORS AND METHODS OF USING THE SAME
[patent_app_type] => utility
[patent_app_number] => 18/443925
[patent_app_country] => US
[patent_app_date] => 2024-02-16
[patent_effective_date] => 0000-00-00
[patent_drawing_sheets_cnt] => 0
[patent_figures_cnt] => 0
[patent_no_of_words] => 56204
[patent_no_of_claims] => 0
[patent_no_of_ind_claims] => 0
[patent_words_short_claim] => 2
[patent_maintenance] => 1
[patent_no_of_assignments] => 0
[patent_current_assignee] =>[type] => publication
[pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18443925
[rel_patent_id] =>[rel_patent_doc_number] =>) 18/443925 | KRAS G12C INHIBITORS AND METHODS OF USING THE SAME | Feb 15, 2024 | Abandoned |
Array
(
[id] => 19233635
[patent_doc_number] => 20240190827
[patent_country] => US
[patent_kind] => A1
[patent_issue_date] => 2024-06-13
[patent_title] => Inhibitors of Rho Associated Coiled-Coil Containing Protein Kinase
[patent_app_type] => utility
[patent_app_number] => 18/434994
[patent_app_country] => US
[patent_app_date] => 2024-02-07
[patent_effective_date] => 0000-00-00
[patent_drawing_sheets_cnt] => 0
[patent_figures_cnt] => 0
[patent_no_of_words] => 22178
[patent_no_of_claims] => 0
[patent_no_of_ind_claims] => -14
[patent_words_short_claim] => 367
[patent_maintenance] => 1
[patent_no_of_assignments] => 0
[patent_current_assignee] =>[type] => publication
[pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18434994
[rel_patent_id] =>[rel_patent_doc_number] =>) 18/434994 | Inhibitors of Rho Associated Coiled-Coil Containing Protein Kinase | Feb 6, 2024 | Pending |
Array
(
[id] => 19180997
[patent_doc_number] => 11987578
[patent_country] => US
[patent_kind] => B1
[patent_issue_date] => 2024-05-21
[patent_title] => 7-(4-((5-(2-chlorobenzylideneamino)-2-thioxo-1,3,4-thiadiazol-3(2H)-yl)methyl)piperazin-1-yl)-1-cyclopropyl-6-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxylic acid as an anti-inflammatory compound
[patent_app_type] => utility
[patent_app_number] => 18/434601
[patent_app_country] => US
[patent_app_date] => 2024-02-06
[patent_effective_date] => 0000-00-00
[patent_drawing_sheets_cnt] => 2
[patent_figures_cnt] => 2
[patent_no_of_words] => 3874
[patent_no_of_claims] => 1
[patent_no_of_ind_claims] => 1
[patent_words_short_claim] => 24
[patent_maintenance] => 1
[patent_no_of_assignments] => 0
[patent_current_assignee] =>[type] => patent
[pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18434601
[rel_patent_id] =>[rel_patent_doc_number] =>) 18/434601 | 7-(4-((5-(2-chlorobenzylideneamino)-2-thioxo-1,3,4-thiadiazol-3(2H)-yl)methyl)piperazin-1-yl)-1-cyclopropyl-6-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxylic acid as an anti-inflammatory compound | Feb 5, 2024 | Issued |
Array
(
[id] => 19667464
[patent_doc_number] => 12180191
[patent_country] => US
[patent_kind] => B1
[patent_issue_date] => 2024-12-31
[patent_title] => 2-[(1H-benzimidazol-2-yl)imino]-5,5-diphenylimidazolidin-4-one as an antimicrobial compound
[patent_app_type] => utility
[patent_app_number] => 18/430400
[patent_app_country] => US
[patent_app_date] => 2024-02-01
[patent_effective_date] => 0000-00-00
[patent_drawing_sheets_cnt] => 2
[patent_figures_cnt] => 2
[patent_no_of_words] => 3995
[patent_no_of_claims] => 1
[patent_no_of_ind_claims] => 1
[patent_words_short_claim] => 113
[patent_maintenance] => 1
[patent_no_of_assignments] => 0
[patent_current_assignee] =>[type] => patent
[pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18430400
[rel_patent_id] =>[rel_patent_doc_number] =>) 18/430400 | 2-[(1H-benzimidazol-2-yl)imino]-5,5-diphenylimidazolidin-4-one as an antimicrobial compound | Jan 31, 2024 | Issued |
Array
(
[id] => 19299896
[patent_doc_number] => 20240228465
[patent_country] => US
[patent_kind] => A1
[patent_issue_date] => 2024-07-11
[patent_title] => SUBSTITUTED PYRIDINE N-OXIDE DERIVATIVES USEFUL AS A FACTOR XIA INHIBITORS
[patent_app_type] => utility
[patent_app_number] => 18/428046
[patent_app_country] => US
[patent_app_date] => 2024-01-31
[patent_effective_date] => 0000-00-00
[patent_drawing_sheets_cnt] => 0
[patent_figures_cnt] => 0
[patent_no_of_words] => 32083
[patent_no_of_claims] => 0
[patent_no_of_ind_claims] => -14
[patent_words_short_claim] => 462
[patent_maintenance] => 1
[patent_no_of_assignments] => 0
[patent_current_assignee] =>[type] => publication
[pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18428046
[rel_patent_id] =>[rel_patent_doc_number] =>) 18/428046 | SUBSTITUTED PYRIDINE N-OXIDE DERIVATIVES USEFUL AS A FACTOR XIA INHIBITORS | Jan 30, 2024 | Abandoned |
Array
(
[id] => 19642866
[patent_doc_number] => 20240417386
[patent_country] => US
[patent_kind] => A1
[patent_issue_date] => 2024-12-19
[patent_title] => INHIBITORS OF RET
[patent_app_type] => utility
[patent_app_number] => 18/422258
[patent_app_country] => US
[patent_app_date] => 2024-01-25
[patent_effective_date] => 0000-00-00
[patent_drawing_sheets_cnt] => 0
[patent_figures_cnt] => 0
[patent_no_of_words] => 17988
[patent_no_of_claims] => 0
[patent_no_of_ind_claims] => -32
[patent_words_short_claim] => 2
[patent_maintenance] => 1
[patent_no_of_assignments] => 0
[patent_current_assignee] =>[type] => publication
[pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18422258
[rel_patent_id] =>[rel_patent_doc_number] =>) 18/422258 | INHIBITORS OF RET | Jan 24, 2024 | Pending |
Array
(
[id] => 19281464
[patent_doc_number] => 20240217938
[patent_country] => US
[patent_kind] => A1
[patent_issue_date] => 2024-07-04
[patent_title] => MORPHIC FORMS OF HEXADECYLOXYPROPYL-PHOSPHONATE ESTERS AND METHODS OF SYNTHESIS THEREOF
[patent_app_type] => utility
[patent_app_number] => 18/414198
[patent_app_country] => US
[patent_app_date] => 2024-01-16
[patent_effective_date] => 0000-00-00
[patent_drawing_sheets_cnt] => 0
[patent_figures_cnt] => 0
[patent_no_of_words] => 32700
[patent_no_of_claims] => 0
[patent_no_of_ind_claims] => -18
[patent_words_short_claim] => 2
[patent_maintenance] => 1
[patent_no_of_assignments] => 0
[patent_current_assignee] =>[type] => publication
[pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18414198
[rel_patent_id] =>[rel_patent_doc_number] =>) 18/414198 | MORPHIC FORMS OF HEXADECYLOXYPROPYL-PHOSPHONATE ESTERS AND METHODS OF SYNTHESIS THEREOF | Jan 15, 2024 | Pending |
Array
(
[id] => 19571766
[patent_doc_number] => 20240376058
[patent_country] => US
[patent_kind] => A1
[patent_issue_date] => 2024-11-14
[patent_title] => GCN2 AND PERK KINASE INHIBITORS AND METHODS OF USE THEREOF
[patent_app_type] => utility
[patent_app_number] => 18/408956
[patent_app_country] => US
[patent_app_date] => 2024-01-10
[patent_effective_date] => 0000-00-00
[patent_drawing_sheets_cnt] => 0
[patent_figures_cnt] => 0
[patent_no_of_words] => 63809
[patent_no_of_claims] => 0
[patent_no_of_ind_claims] => -26
[patent_words_short_claim] => 2
[patent_maintenance] => 1
[patent_no_of_assignments] => 0
[patent_current_assignee] =>[type] => publication
[pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18408956
[rel_patent_id] =>[rel_patent_doc_number] =>) 18/408956 | GCN2 AND PERK KINASE INHIBITORS AND METHODS OF USE THEREOF | Jan 9, 2024 | Pending |
Array
(
[id] => 19112675
[patent_doc_number] => 20240124425
[patent_country] => US
[patent_kind] => A1
[patent_issue_date] => 2024-04-18
[patent_title] => SOLID STATE FORMS OF BELUMOSUDIL AND BELUMOSUDIL SALTS
[patent_app_type] => utility
[patent_app_number] => 18/393915
[patent_app_country] => US
[patent_app_date] => 2023-12-22
[patent_effective_date] => 0000-00-00
[patent_drawing_sheets_cnt] => 0
[patent_figures_cnt] => 0
[patent_no_of_words] => 16944
[patent_no_of_claims] => 0
[patent_no_of_ind_claims] => -15
[patent_words_short_claim] => 123
[patent_maintenance] => 1
[patent_no_of_assignments] => 0
[patent_current_assignee] =>[type] => publication
[pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18393915
[rel_patent_id] =>[rel_patent_doc_number] =>) 18/393915 | Solid state forms of Belumosudil and Belumosudil salts | Dec 21, 2023 | Issued |
Array
(
[id] => 19403566
[patent_doc_number] => 20240287077
[patent_country] => US
[patent_kind] => A1
[patent_issue_date] => 2024-08-29
[patent_title] => PYRAZOLOPYRIMIDINE COMPOUNDS
[patent_app_type] => utility
[patent_app_number] => 18/391047
[patent_app_country] => US
[patent_app_date] => 2023-12-20
[patent_effective_date] => 0000-00-00
[patent_drawing_sheets_cnt] => 0
[patent_figures_cnt] => 0
[patent_no_of_words] => 12996
[patent_no_of_claims] => 0
[patent_no_of_ind_claims] => -8
[patent_words_short_claim] => 65
[patent_maintenance] => 1
[patent_no_of_assignments] => 0
[patent_current_assignee] =>[type] => publication
[pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18391047
[rel_patent_id] =>[rel_patent_doc_number] =>) 18/391047 | PYRAZOLOPYRIMIDINE COMPOUNDS | Dec 19, 2023 | Abandoned |
Array
(
[id] => 19165789
[patent_doc_number] => 11981675
[patent_country] => US
[patent_kind] => B1
[patent_issue_date] => 2024-05-14
[patent_title] => Pyrrolo[3,2-C]quinoline-2,3-dione compounds as CK2 inhibitors
[patent_app_type] => utility
[patent_app_number] => 18/536912
[patent_app_country] => US
[patent_app_date] => 2023-12-12
[patent_effective_date] => 0000-00-00
[patent_drawing_sheets_cnt] => 0
[patent_figures_cnt] => 0
[patent_no_of_words] => 9462
[patent_no_of_claims] => 17
[patent_no_of_ind_claims] => 3
[patent_words_short_claim] => 66
[patent_maintenance] => 1
[patent_no_of_assignments] => 0
[patent_current_assignee] =>[type] => patent
[pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18536912
[rel_patent_id] =>[rel_patent_doc_number] =>) 18/536912 | Pyrrolo[3,2-C]quinoline-2,3-dione compounds as CK2 inhibitors | Dec 11, 2023 | Issued |
Array
(
[id] => 19105770
[patent_doc_number] => 11958851
[patent_country] => US
[patent_kind] => B1
[patent_issue_date] => 2024-04-16
[patent_title] => Pyrrolo[3,2-c]quinoline compounds as CK2 inhibitors
[patent_app_type] => utility
[patent_app_number] => 18/533067
[patent_app_country] => US
[patent_app_date] => 2023-12-07
[patent_effective_date] => 0000-00-00
[patent_drawing_sheets_cnt] => 0
[patent_figures_cnt] => 0
[patent_no_of_words] => 9694
[patent_no_of_claims] => 10
[patent_no_of_ind_claims] => 1
[patent_words_short_claim] => 391
[patent_maintenance] => 1
[patent_no_of_assignments] => 0
[patent_current_assignee] =>[type] => patent
[pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18533067
[rel_patent_id] =>[rel_patent_doc_number] =>) 18/533067 | Pyrrolo[3,2-c]quinoline compounds as CK2 inhibitors | Dec 6, 2023 | Issued |
Array
(
[id] => 19135566
[patent_doc_number] => 11970496
[patent_country] => US
[patent_kind] => B1
[patent_issue_date] => 2024-04-30
[patent_title] => Pyrrolo[3,2-c]quinoline compounds as CK2 inhibitors
[patent_app_type] => utility
[patent_app_number] => 18/533073
[patent_app_country] => US
[patent_app_date] => 2023-12-07
[patent_effective_date] => 0000-00-00
[patent_drawing_sheets_cnt] => 0
[patent_figures_cnt] => 0
[patent_no_of_words] => 9698
[patent_no_of_claims] => 11
[patent_no_of_ind_claims] => 3
[patent_words_short_claim] => 101
[patent_maintenance] => 1
[patent_no_of_assignments] => 0
[patent_current_assignee] =>[type] => patent
[pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18533073
[rel_patent_id] =>[rel_patent_doc_number] =>) 18/533073 | Pyrrolo[3,2-c]quinoline compounds as CK2 inhibitors | Dec 6, 2023 | Issued |
Array
(
[id] => 19157605
[patent_doc_number] => 20240150312
[patent_country] => US
[patent_kind] => A1
[patent_issue_date] => 2024-05-09
[patent_title] => PYRAZINE COMPOUND
[patent_app_type] => utility
[patent_app_number] => 18/532293
[patent_app_country] => US
[patent_app_date] => 2023-12-07
[patent_effective_date] => 0000-00-00
[patent_drawing_sheets_cnt] => 0
[patent_figures_cnt] => 0
[patent_no_of_words] => 51784
[patent_no_of_claims] => 0
[patent_no_of_ind_claims] => 0
[patent_words_short_claim] => 221
[patent_maintenance] => 1
[patent_no_of_assignments] => 0
[patent_current_assignee] =>[type] => publication
[pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18532293
[rel_patent_id] =>[rel_patent_doc_number] =>) 18/532293 | PYRAZINE COMPOUND | Dec 6, 2023 | Abandoned |
Array
(
[id] => 19543059
[patent_doc_number] => 20240360095
[patent_country] => US
[patent_kind] => A1
[patent_issue_date] => 2024-10-31
[patent_title] => NOVEL KINASE MODULATORS
[patent_app_type] => utility
[patent_app_number] => 18/508085
[patent_app_country] => US
[patent_app_date] => 2023-11-13
[patent_effective_date] => 0000-00-00
[patent_drawing_sheets_cnt] => 0
[patent_figures_cnt] => 0
[patent_no_of_words] => 75212
[patent_no_of_claims] => 0
[patent_no_of_ind_claims] => -23
[patent_words_short_claim] => 2
[patent_maintenance] => 1
[patent_no_of_assignments] => 0
[patent_current_assignee] =>[type] => publication
[pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18508085
[rel_patent_id] =>[rel_patent_doc_number] =>) 18/508085 | NOVEL KINASE MODULATORS | Nov 12, 2023 | Pending |
| 18/388734 | 5-(SUBSTITUTEDPHENYL)-7-THIOXO-7,8-DIHYDROPYRIMIDO[4,5- d]PYRIMIDINE-2,4(1H,3H)-DIONE ANALOGUES AS ANTIBACTERIAL AGENTS | Nov 9, 2023 | |
Array
(
[id] => 19135542
[patent_doc_number] => 11970472
[patent_country] => US
[patent_kind] => B1
[patent_issue_date] => 2024-04-30
[patent_title] => 5-((2-isopropyl-5-methylphenoxy)methyl)-3-(naphthalen-1-yl)-1,2,4-oxadiazole as an anti-cancer and antimicrobial compound
[patent_app_type] => utility
[patent_app_number] => 18/386545
[patent_app_country] => US
[patent_app_date] => 2023-11-02
[patent_effective_date] => 0000-00-00
[patent_drawing_sheets_cnt] => 0
[patent_figures_cnt] => 0
[patent_no_of_words] => 4475
[patent_no_of_claims] => 10
[patent_no_of_ind_claims] => 1
[patent_words_short_claim] => 8
[patent_maintenance] => 1
[patent_no_of_assignments] => 0
[patent_current_assignee] =>[type] => patent
[pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18386545
[rel_patent_id] =>[rel_patent_doc_number] =>) 18/386545 | 5-((2-isopropyl-5-methylphenoxy)methyl)-3-(naphthalen-1-yl)-1,2,4-oxadiazole as an anti-cancer and antimicrobial compound | Nov 1, 2023 | Issued |
Array
(
[id] => 20414117
[patent_doc_number] => 12497387
[patent_country] => US
[patent_kind] => B2
[patent_issue_date] => 2025-12-16
[patent_title] => Process for the preparation of pyrimidinyl-4-aminopyrazole compounds
[patent_app_type] => utility
[patent_app_number] => 18/384080
[patent_app_country] => US
[patent_app_date] => 2023-10-26
[patent_effective_date] => 0000-00-00
[patent_drawing_sheets_cnt] => 0
[patent_figures_cnt] => 0
[patent_no_of_words] => 1730
[patent_no_of_claims] => 5
[patent_no_of_ind_claims] => 1
[patent_words_short_claim] => 247
[patent_maintenance] => 1
[patent_no_of_assignments] => 0
[patent_current_assignee] =>[type] => patent
[pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18384080
[rel_patent_id] =>[rel_patent_doc_number] =>) 18/384080 | Process for the preparation of pyrimidinyl-4-aminopyrazole compounds | Oct 25, 2023 | Issued |