Search

Bruck Kifle

Examiner (ID: 2332)

Most Active Art Unit
1624
Art Unit(s)
1202, 1624, 1611, 1622
Total Applications
3434
Issued Applications
2601
Pending Applications
222
Abandoned Applications
651

Applications

Application numberTitle of the applicationFiling DateStatus
Array ( [id] => 14171645 [patent_doc_number] => 10259817 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2019-04-16 [patent_title] => Crystal (6S,9aS)-N-benzyl-8-({6-[3-(4-ethylpiperazin-1-yl)azetidin-1-yl]pyridin-2-yl}methyl)-6-(2-fluoro-4-hydroxybenzyl)-4,7-dioxo-2-(prop-2-en-1-yl)hexahydro-2H-pyrazino[2,1-c][1,2,4]triazine-1(6H)-carboxamide [patent_app_type] => utility [patent_app_number] => 15/577858 [patent_app_country] => US [patent_app_date] => 2016-06-21 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 6 [patent_figures_cnt] => 6 [patent_no_of_words] => 8765 [patent_no_of_claims] => 8 [patent_no_of_ind_claims] => 2 [patent_words_short_claim] => 25 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 15577858 [rel_patent_id] =>[rel_patent_doc_number] =>)
15/577858
Crystal (6S,9aS)-N-benzyl-8-({6-[3-(4-ethylpiperazin-1-yl)azetidin-1-yl]pyridin-2-yl}methyl)-6-(2-fluoro-4-hydroxybenzyl)-4,7-dioxo-2-(prop-2-en-1-yl)hexahydro-2H-pyrazino[2,1-c][1,2,4]triazine-1(6H)-carboxamide Jun 20, 2016 Issued
Array ( [id] => 16406699 [patent_doc_number] => 10815242 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2020-10-27 [patent_title] => Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment [patent_app_type] => utility [patent_app_number] => 15/736697 [patent_app_country] => US [patent_app_date] => 2016-06-17 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 10 [patent_figures_cnt] => 10 [patent_no_of_words] => 70144 [patent_no_of_claims] => 10 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 433 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 15736697 [rel_patent_id] =>[rel_patent_doc_number] =>)
15/736697
Benzodiazepine derivatives, compositions, and methods for treating cognitive impairment Jun 16, 2016 Issued
Array ( [id] => 12884692 [patent_doc_number] => 20180186739 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2018-07-05 [patent_title] => SPIRO[CYCLOBUTANE-1,3'-INDOLIN]-2'-ONE DERIVATIVES AS BROMODOMAIN INHIBITORS [patent_app_type] => utility [patent_app_number] => 15/736450 [patent_app_country] => US [patent_app_date] => 2016-06-15 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 44718 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -31 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 15736450 [rel_patent_id] =>[rel_patent_doc_number] =>)
15/736450
Spiro[cyclobutane-1,3'-indolin]-2'-one derivatives as bromodomain inhibitors Jun 14, 2016 Issued
Array ( [id] => 11749303 [patent_doc_number] => 09707301 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2017-07-18 [patent_title] => 'Pyrrolobenzodiazepines and targeted conjugates' [patent_app_type] => utility [patent_app_number] => 15/182649 [patent_app_country] => US [patent_app_date] => 2016-06-15 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 1 [patent_figures_cnt] => 2 [patent_no_of_words] => 28781 [patent_no_of_claims] => 10 [patent_no_of_ind_claims] => 2 [patent_words_short_claim] => 26 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 15182649 [rel_patent_id] =>[rel_patent_doc_number] =>)
15/182649
Pyrrolobenzodiazepines and targeted conjugates Jun 14, 2016 Issued
Array ( [id] => 15696685 [patent_doc_number] => 10604509 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2020-03-31 [patent_title] => Nrf2 regulators [patent_app_type] => utility [patent_app_number] => 15/736075 [patent_app_country] => US [patent_app_date] => 2016-06-15 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 99433 [patent_no_of_claims] => 26 [patent_no_of_ind_claims] => 5 [patent_words_short_claim] => 7 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 15736075 [rel_patent_id] =>[rel_patent_doc_number] =>)
15/736075
Nrf2 regulators Jun 14, 2016 Issued
Array ( [id] => 11092270 [patent_doc_number] => 20160289239 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2016-10-06 [patent_title] => 'PYRROLOBENZODIAZEPINES AND TARGETED CONJUGATES' [patent_app_type] => utility [patent_app_number] => 15/181900 [patent_app_country] => US [patent_app_date] => 2016-06-14 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 1 [patent_figures_cnt] => 1 [patent_no_of_words] => 27654 [patent_no_of_claims] => 11 [patent_no_of_ind_claims] => 2 [patent_words_short_claim] => 0 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 15181900 [rel_patent_id] =>[rel_patent_doc_number] =>)
15/181900
Pyrrolobenzodiazepines and targeted conjugates Jun 13, 2016 Issued
Array ( [id] => 11364051 [patent_doc_number] => 20170002033 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2017-01-05 [patent_title] => 'ACYCLIC NUCLEOSIDE PHOSPHONATE DIESTERS' [patent_app_type] => utility [patent_app_number] => 15/179209 [patent_app_country] => US [patent_app_date] => 2016-06-10 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 1 [patent_figures_cnt] => 1 [patent_no_of_words] => 37109 [patent_no_of_claims] => 28 [patent_no_of_ind_claims] => 6 [patent_words_short_claim] => 0 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 15179209 [rel_patent_id] =>[rel_patent_doc_number] =>)
15/179209
Acyclic nucleoside phosphonate diesters Jun 9, 2016 Issued
Array ( [id] => 12408306 [patent_doc_number] => 09969700 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2018-05-15 [patent_title] => P2X4 receptor antagonist [patent_app_type] => utility [patent_app_number] => 15/176857 [patent_app_country] => US [patent_app_date] => 2016-06-08 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 40489 [patent_no_of_claims] => 11 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 1562 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 15176857 [rel_patent_id] =>[rel_patent_doc_number] =>)
15/176857
P2X4 receptor antagonist Jun 7, 2016 Issued
Array ( [id] => 12808828 [patent_doc_number] => 20180161446 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2018-06-14 [patent_title] => ANTIBODY DRUG CONJUGATE, INTERMEDIATE, PREPARATION METHOD, PHARMACEUTICAL COMPOSITION AND USES THEREOF [patent_app_type] => utility [patent_app_number] => 15/580895 [patent_app_country] => US [patent_app_date] => 2016-06-08 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 34462 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -17 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 15580895 [rel_patent_id] =>[rel_patent_doc_number] =>)
15/580895
Antibody drug conjugate, intermediate, preparation method, pharmaceutical composition and uses thereof Jun 7, 2016 Issued
Array ( [id] => 11083697 [patent_doc_number] => 20160280662 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2016-09-29 [patent_title] => '5-FLUORO-4-IMINO-3-(ALKYL/SUBSTITUTED ALKYL)-1-(ARYLSULFONYL)-3,4-DIHYDROPYRIMIDIN-2(1H)-ONE AND PROCESSES FOR THEIR PREPARATION' [patent_app_type] => utility [patent_app_number] => 15/173493 [patent_app_country] => US [patent_app_date] => 2016-06-03 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 3028 [patent_no_of_claims] => 17 [patent_no_of_ind_claims] => 2 [patent_words_short_claim] => 0 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 15173493 [rel_patent_id] =>[rel_patent_doc_number] =>)
15/173493
5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1 H)-one and processes for their preparation Jun 2, 2016 Issued
Array ( [id] => 12812917 [patent_doc_number] => 20180162809 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2018-06-14 [patent_title] => ROR GAMMA (RORY) MODULATORS [patent_app_type] => utility [patent_app_number] => 15/579075 [patent_app_country] => US [patent_app_date] => 2016-06-03 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 8178 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -16 [patent_words_short_claim] => 213 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 15579075 [rel_patent_id] =>[rel_patent_doc_number] =>)
15/579075
ROR gamma (RORy) modulators Jun 2, 2016 Issued
Array ( [id] => 15483067 [patent_doc_number] => 10556866 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2020-02-11 [patent_title] => ROR gamma (RORg) modulators [patent_app_type] => utility [patent_app_number] => 15/579164 [patent_app_country] => US [patent_app_date] => 2016-06-03 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 13008 [patent_no_of_claims] => 6 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 395 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 15579164 [rel_patent_id] =>[rel_patent_doc_number] =>)
15/579164
ROR gamma (RORg) modulators Jun 2, 2016 Issued
Array ( [id] => 11083698 [patent_doc_number] => 20160280663 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2016-09-29 [patent_title] => '5-FLUORO-4-IMINO-3-(ALKYL/SUBSTITUTED ALKYL)-1-(ARYLSULFONYL)-3,4-DIHYDROPYRIMIDIN-2(1H)-ONE AND PROCESSES FOR THEIR PREPARATION' [patent_app_type] => utility [patent_app_number] => 15/173529 [patent_app_country] => US [patent_app_date] => 2016-06-03 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 3033 [patent_no_of_claims] => 17 [patent_no_of_ind_claims] => 2 [patent_words_short_claim] => 0 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 15173529 [rel_patent_id] =>[rel_patent_doc_number] =>)
15/173529
5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1H)-one and processes for their preparation Jun 2, 2016 Issued
Array ( [id] => 12812950 [patent_doc_number] => 20180162820 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2018-06-14 [patent_title] => NEW METHOD FOR THE PREPARATION OF HIGHLY PURE IVABRADINE BASE AND SALTS THEREOF [patent_app_type] => utility [patent_app_number] => 15/735172 [patent_app_country] => US [patent_app_date] => 2016-06-02 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 3877 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -15 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 15735172 [rel_patent_id] =>[rel_patent_doc_number] =>)
15/735172
Method for the preparation of highly pure ivabradine base and salts thereof Jun 1, 2016 Issued
Array ( [id] => 11311680 [patent_doc_number] => 20160347790 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2016-12-01 [patent_title] => 'SYNTHESIS OF SYRBACTIN PROTEASOME INHIBITORS' [patent_app_type] => utility [patent_app_number] => 15/171513 [patent_app_country] => US [patent_app_date] => 2016-06-02 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 2 [patent_figures_cnt] => 2 [patent_no_of_words] => 9835 [patent_no_of_claims] => 21 [patent_no_of_ind_claims] => 4 [patent_words_short_claim] => 0 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 15171513 [rel_patent_id] =>[rel_patent_doc_number] =>)
15/171513
Synthesis of syrbactin proteasome inhibitors Jun 1, 2016 Issued
Array ( [id] => 12837067 [patent_doc_number] => 20180170862 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2018-06-21 [patent_title] => PROTEIN TYROSINE PHOSPHATASES OR SHP2 INHIBITORS AND USES THEREOF [patent_app_type] => utility [patent_app_number] => 15/577417 [patent_app_country] => US [patent_app_date] => 2016-06-01 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 22887 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -14 [patent_words_short_claim] => 136 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 15577417 [rel_patent_id] =>[rel_patent_doc_number] =>)
15/577417
Protein tyrosine phosphatases or SHP2 inhibitors and uses thereof May 31, 2016 Issued
Array ( [id] => 12837064 [patent_doc_number] => 20180170861 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2018-06-21 [patent_title] => SMALL MOLECULE INHIBITORS OF PROTEIN TYROSINE PHOSPHATASES AND USED THEREOF [patent_app_type] => utility [patent_app_number] => 15/577398 [patent_app_country] => US [patent_app_date] => 2016-06-01 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 23021 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -16 [patent_words_short_claim] => 80 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 15577398 [rel_patent_id] =>[rel_patent_doc_number] =>)
15/577398
Small molecule inhibitors of protein tyrosine phosphatases and uses thereof May 31, 2016 Issued
Array ( [id] => 11121899 [patent_doc_number] => 20160318873 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2016-11-03 [patent_title] => 'POLYMORPHIC FORMS OF IVABRADINE HYDROCHLORIDE' [patent_app_type] => utility [patent_app_number] => 15/168880 [patent_app_country] => US [patent_app_date] => 2016-05-31 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 3 [patent_figures_cnt] => 3 [patent_no_of_words] => 5950 [patent_no_of_claims] => 11 [patent_no_of_ind_claims] => 3 [patent_words_short_claim] => 0 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 15168880 [rel_patent_id] =>[rel_patent_doc_number] =>)
15/168880
Polymorphic forms of ivabradine hydrochloride May 30, 2016 Issued
Array ( [id] => 13763405 [patent_doc_number] => 10174037 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2019-01-08 [patent_title] => Dihydropyrazolopyrimidinone compounds as PDE2 inhibitors [patent_app_type] => utility [patent_app_number] => 15/576351 [patent_app_country] => US [patent_app_date] => 2016-05-31 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 43918 [patent_no_of_claims] => 19 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 189 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 15576351 [rel_patent_id] =>[rel_patent_doc_number] =>)
15/576351
Dihydropyrazolopyrimidinone compounds as PDE2 inhibitors May 30, 2016 Issued
Array ( [id] => 15193803 [patent_doc_number] => 10494380 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2019-12-03 [patent_title] => Nitrogen-containing tricyclic derivatives having HIV replication inhibitory activity [patent_app_type] => utility [patent_app_number] => 15/577795 [patent_app_country] => US [patent_app_date] => 2016-05-27 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 74375 [patent_no_of_claims] => 37 [patent_no_of_ind_claims] => 6 [patent_words_short_claim] => 12 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 15577795 [rel_patent_id] =>[rel_patent_doc_number] =>)
15/577795
Nitrogen-containing tricyclic derivatives having HIV replication inhibitory activity May 26, 2016 Issued
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