Search

Douglas M. Willis

Examiner (ID: 5249, Phone: (571)270-5757 , Office: P/1624 )

Most Active Art Unit
1624
Art Unit(s)
1624
Total Applications
2485
Issued Applications
1796
Pending Applications
148
Abandoned Applications
577

Applications

Application numberTitle of the applicationFiling DateStatus
Array ( [id] => 17776526 [patent_doc_number] => 20220242875 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-08-04 [patent_title] => INHIBITORS OF KRAS G12C [patent_app_type] => utility [patent_app_number] => 17/716707 [patent_app_country] => US [patent_app_date] => 2022-04-08 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 57711 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -12 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17716707 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/716707
Substituted piperazines as inhibitors of KRAS G12C Apr 7, 2022 Issued
Array ( [id] => 17776526 [patent_doc_number] => 20220242875 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-08-04 [patent_title] => INHIBITORS OF KRAS G12C [patent_app_type] => utility [patent_app_number] => 17/716707 [patent_app_country] => US [patent_app_date] => 2022-04-08 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 57711 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -12 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17716707 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/716707
Substituted piperazines as inhibitors of KRAS G12C Apr 7, 2022 Issued
Array ( [id] => 17761423 [patent_doc_number] => 20220235035 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-07-28 [patent_title] => TYK2 INHIBITORS AND USES THEREOF [patent_app_type] => utility [patent_app_number] => 17/713646 [patent_app_country] => US [patent_app_date] => 2022-04-05 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 86920 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => 0 [patent_words_short_claim] => 11 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17713646 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/713646
Substituted 1,2,4-triazoles as intermediates in the synthesis of TYK2 inhibitors Apr 4, 2022 Issued
Array ( [id] => 17749571 [patent_doc_number] => 20220227775 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-07-21 [patent_title] => 1H-PYRAZOLO[4,3-H]QUINAZOLINE COMPOUND SERVING AS PROTEIN KINASE INHIBITOR [patent_app_type] => utility [patent_app_number] => 17/711535 [patent_app_country] => US [patent_app_date] => 2022-04-01 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 24714 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -17 [patent_words_short_claim] => 95 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17711535 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/711535
Substituted pyrazolo[4,3-H]quinazolines as protein kinase inhibitors Mar 31, 2022 Issued
Array ( [id] => 18004929 [patent_doc_number] => 20220363695 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-11-17 [patent_title] => HPK1 ANTAGONISTS AND USES THEREOF [patent_app_type] => utility [patent_app_number] => 17/656924 [patent_app_country] => US [patent_app_date] => 2022-03-29 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 45877 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -19 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17656924 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/656924
Substituted pyrrolo[3,4-c]pyridines as HPK1 antagonists Mar 28, 2022 Issued
Array ( [id] => 18093079 [patent_doc_number] => 20220411420 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-12-29 [patent_title] => PYRROLOPYRIMIDINE DERIVATIVE HAVING ECTONUCLEOTIDE PYROPHOSPHATASE-PHOSPHODIESTERASE INHIBITORY ACTIVITY AND USE THEREOF [patent_app_type] => utility [patent_app_number] => 17/706628 [patent_app_country] => US [patent_app_date] => 2022-03-29 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 21516 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -13 [patent_words_short_claim] => 754 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17706628 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/706628
Substituted pyrrolo[2,3-d]pyrimidines having ectonucleotide pyrophosphatase-phosphodiesterase inhibitory activity Mar 28, 2022 Issued
Array ( [id] => 18987725 [patent_doc_number] => 20240059694 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-02-22 [patent_title] => COMPOUND CONTAINING 1,3-BENZODIOXOL STRUCTURE AND PREPARATION METHOD AND USE THEREOF [patent_app_type] => utility [patent_app_number] => 18/257027 [patent_app_country] => US [patent_app_date] => 2022-03-24 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 18742 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -14 [patent_words_short_claim] => 164 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18257027 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/257027
COMPOUND CONTAINING 1,3-BENZODIOXOL STRUCTURE AND PREPARATION METHOD AND USE THEREOF Mar 23, 2022 Pending
Array ( [id] => 17734655 [patent_doc_number] => 20220220114 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-07-14 [patent_title] => PHOSPHODIESTERASE INHIBITORS AND USE [patent_app_type] => utility [patent_app_number] => 17/702704 [patent_app_country] => US [patent_app_date] => 2022-03-23 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 31823 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -29 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17702704 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/702704
Substituted imidazo[4,5-c][1,8]naphthyridines as phosphodiesterase inhibitors Mar 22, 2022 Issued
Array ( [id] => 17734659 [patent_doc_number] => 20220220118 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-07-14 [patent_title] => ION CHANNEL MODULATORS [patent_app_type] => utility [patent_app_number] => 17/702518 [patent_app_country] => US [patent_app_date] => 2022-03-23 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 52333 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -13 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17702518 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/702518
3-(ethoxydifluoromethyl)-6-(5-fluoro-6-(2,2,2-trifluoroethoxy)pyridin-3-yl)-[1,2,4]triazolo[4,3-a]pyridine as an ion channel modulator Mar 22, 2022 Issued
Array ( [id] => 19397080 [patent_doc_number] => 12071421 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2024-08-27 [patent_title] => Process for the synthesis of substituted chloromethyl dialkylphosphates [patent_app_type] => utility [patent_app_number] => 17/699522 [patent_app_country] => US [patent_app_date] => 2022-03-21 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 1 [patent_figures_cnt] => 1 [patent_no_of_words] => 15014 [patent_no_of_claims] => 3 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 818 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17699522 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/699522
Process for the synthesis of substituted chloromethyl dialkylphosphates Mar 20, 2022 Issued
Array ( [id] => 18278389 [patent_doc_number] => 20230093861 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2023-03-30 [patent_title] => RAPAMYCIN ANALOGS AS MTOR INHIBITORS [patent_app_type] => utility [patent_app_number] => 17/693225 [patent_app_country] => US [patent_app_date] => 2022-03-11 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 66558 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -29 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17693225 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/693225
RAPAMYCIN ANALOGS AS MTOR INHIBITORS Mar 10, 2022 Abandoned
Array ( [id] => 19332530 [patent_doc_number] => 20240246960 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-07-25 [patent_title] => 7-Morpholino-L,6-Naphthyridin-5-yl Derivatives and Pharmaceutical Compositions Thereof Useful as DNA-PK Inhibitor [patent_app_type] => utility [patent_app_number] => 18/279377 [patent_app_country] => US [patent_app_date] => 2022-03-10 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 69274 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -38 [patent_words_short_claim] => 19 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18279377 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/279377
7-Morpholino-L,6-Naphthyridin-5-yl Derivatives and Pharmaceutical Compositions Thereof Useful as DNA-PK Inhibitor Mar 9, 2022 Pending
Array ( [id] => 17866951 [patent_doc_number] => 20220289686 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-09-15 [patent_title] => COMPOSITIONS OF NRF2 INHIBITING AGENTS AND METHODS OF USE THEREOF [patent_app_type] => utility [patent_app_number] => 17/690826 [patent_app_country] => US [patent_app_date] => 2022-03-09 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 22126 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -19 [patent_words_short_claim] => 93 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17690826 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/690826
COMPOSITIONS OF NRF2 INHIBITING AGENTS AND METHODS OF USE THEREOF Mar 8, 2022 Abandoned
Array ( [id] => 17720391 [patent_doc_number] => 20220213111 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-07-07 [patent_title] => SUBSTITUTED HETEROCYCLES AS CYCLIC TREX1 INHIBITORS [patent_app_type] => utility [patent_app_number] => 17/653904 [patent_app_country] => US [patent_app_date] => 2022-03-08 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 18556 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -11 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17653904 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/653904
SUBSTITUTED HETEROCYCLES AS CYCLIC TREX1 INHIBITORS Mar 7, 2022 Abandoned
Array ( [id] => 19423697 [patent_doc_number] => 12083088 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2024-09-10 [patent_title] => Substituted esters containing polyols and saccharides for treating hepatotoxicity and fatty liver diseases [patent_app_type] => utility [patent_app_number] => 17/686013 [patent_app_country] => US [patent_app_date] => 2022-03-03 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 6 [patent_figures_cnt] => 6 [patent_no_of_words] => 18876 [patent_no_of_claims] => 81 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 207 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17686013 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/686013
Substituted esters containing polyols and saccharides for treating hepatotoxicity and fatty liver diseases Mar 2, 2022 Issued
Array ( [id] => 18225366 [patent_doc_number] => 20230064360 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2023-03-02 [patent_title] => HETEROCYCLES AND USES THEREOF [patent_app_type] => utility [patent_app_number] => 17/685370 [patent_app_country] => US [patent_app_date] => 2022-03-02 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 193002 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -25 [patent_words_short_claim] => 13 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17685370 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/685370
Substituted pyrido[2,3-d]pyrimidines as inhibitors of Ras pathway signaling Mar 1, 2022 Issued
Array ( [id] => 18321342 [patent_doc_number] => 20230119470 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2023-04-20 [patent_title] => PYRAZINO[2,3-b]PYRAZINE mTOR KINASE INHIBITORS FOR ONCOLOGY INDICATIONS AND DISEASES ASSOCIATED WITH THE mTOR/PI3K/AKT PATHWAY [patent_app_type] => utility [patent_app_number] => 17/681645 [patent_app_country] => US [patent_app_date] => 2022-02-25 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 39837 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => 0 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17681645 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/681645
PYRAZINO[2,3-b]PYRAZINE mTOR KINASE INHIBITORS FOR ONCOLOGY INDICATIONS AND DISEASES ASSOCIATED WITH THE mTOR/PI3K/AKT PATHWAY Feb 24, 2022 Abandoned
Array ( [id] => 19359696 [patent_doc_number] => 20240261730 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-08-08 [patent_title] => METHOD FOR PRODUCING 2-FURONITRILE AND METHOD FOR PRODUCING CARBONIC ACID ESTER [patent_app_type] => utility [patent_app_number] => 18/276778 [patent_app_country] => US [patent_app_date] => 2022-02-24 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 5451 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -9 [patent_words_short_claim] => 28 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18276778 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/276778
METHOD FOR PRODUCING 2-FURONITRILE AND METHOD FOR PRODUCING CARBONIC ACID ESTER Feb 23, 2022 Pending
Array ( [id] => 17657017 [patent_doc_number] => 20220177482 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-06-09 [patent_title] => PROCESS FOR THE PREPARATION OF N-((1R,2S,5R)-5-(TERT-BUTYLAMINO)-2-((S)-3-(7-TERT-BUTYLPYRAZOLO[1,5-A][1,3,5]TRIAZIN-4-YLAMINO)-2-OXOPYRROLIDIN-1-YL)CYCLOHEXYL)ACETAMIDE [patent_app_type] => utility [patent_app_number] => 17/677312 [patent_app_country] => US [patent_app_date] => 2022-02-22 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 7207 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => 0 [patent_words_short_claim] => 24 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17677312 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/677312
PROCESS FOR THE PREPARATION OF N-((1R,2S,5R)-5-(TERT-BUTYLAMINO)-2-((S)-3-(7-TERT-BUTYLPYRAZOLO[1,5-A][1,3,5]TRIAZIN-4-YLAMINO)-2-OXOPYRROLIDIN-1-YL)CYCLOHEXYL)ACETAMIDE Feb 21, 2022 Abandoned
Array ( [id] => 18987727 [patent_doc_number] => 20240059696 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-02-22 [patent_title] => PROCESS FOR PREPARING HIGH PURITY DEGREE LAROTRECTINIB [patent_app_type] => utility [patent_app_number] => 18/270781 [patent_app_country] => US [patent_app_date] => 2022-02-18 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 2408 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -6 [patent_words_short_claim] => 4 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18270781 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/270781
PROCESS FOR PREPARING HIGH PURITY DEGREE LAROTRECTINIB Feb 17, 2022 Pending
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