Search

Douglas M. Willis

Examiner (ID: 5249, Phone: (571)270-5757 , Office: P/1624 )

Most Active Art Unit
1624
Art Unit(s)
1624
Total Applications
2485
Issued Applications
1796
Pending Applications
148
Abandoned Applications
577

Applications

Application numberTitle of the applicationFiling DateStatus
Array ( [id] => 17015198 [patent_doc_number] => 11084825 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2021-08-10 [patent_title] => Substituted pyridines as irreversible inhibitors of menin-MLL interaction [patent_app_type] => utility [patent_app_number] => 16/732226 [patent_app_country] => US [patent_app_date] => 2019-12-31 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 5 [patent_figures_cnt] => 8 [patent_no_of_words] => 57921 [patent_no_of_claims] => 26 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 668 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16732226 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/732226
Substituted pyridines as irreversible inhibitors of menin-MLL interaction Dec 30, 2019 Issued
Array ( [id] => 16190739 [patent_doc_number] => 20200231588 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2020-07-23 [patent_title] => Bicyclic Heteroaryl Compounds [patent_app_type] => utility [patent_app_number] => 16/722881 [patent_app_country] => US [patent_app_date] => 2019-12-20 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 22913 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -8 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16722881 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/722881
Bicyclic Heteroaryl Compounds Dec 19, 2019 Abandoned
Array ( [id] => 16572881 [patent_doc_number] => 10894794 [patent_country] => US [patent_kind] => B1 [patent_issue_date] => 2021-01-19 [patent_title] => Substituted [1,2,4]triazolo[4,3-a]pyrazines as antidiabetics [patent_app_type] => utility [patent_app_number] => 16/719014 [patent_app_country] => US [patent_app_date] => 2019-12-18 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 18 [patent_figures_cnt] => 31 [patent_no_of_words] => 8664 [patent_no_of_claims] => 16 [patent_no_of_ind_claims] => 3 [patent_words_short_claim] => 15 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16719014 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/719014
Substituted [1,2,4]triazolo[4,3-a]pyrazines as antidiabetics Dec 17, 2019 Issued
Array ( [id] => 15768725 [patent_doc_number] => 20200115380 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2020-04-16 [patent_title] => SUBSTITUTED HETEROCYCLE FUSED GAMMA-CARBOLINES SYNTHESIS [patent_app_type] => utility [patent_app_number] => 16/711790 [patent_app_country] => US [patent_app_date] => 2019-12-12 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 19976 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -7 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16711790 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/711790
Preparation of certain substituted 1H-pyrido[3',4':4,5]pyrrolo[1,2,3-de]quinoxalines and pharmaceutically acceptable salts thereof Dec 11, 2019 Issued
Array ( [id] => 16072213 [patent_doc_number] => 20200190093 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2020-06-18 [patent_title] => SUBSTITUTED XANTHINE DERIVATIVES [patent_app_type] => utility [patent_app_number] => 16/710887 [patent_app_country] => US [patent_app_date] => 2019-12-11 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 18397 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -13 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16710887 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/710887
Substituted xanthines as inhibitors of transient receptor potential cation channel subfamily c, member 5 activity Dec 10, 2019 Issued
Array ( [id] => 17428324 [patent_doc_number] => 20220056032 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-02-24 [patent_title] => SUBSTITUTED XANTHINE DERIVATIVES [patent_app_type] => utility [patent_app_number] => 17/312831 [patent_app_country] => US [patent_app_date] => 2019-12-10 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 6672 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -14 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17312831 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/312831
Substituted xanthines as modulators of TRPC5 activity Dec 9, 2019 Issued
Array ( [id] => 16072211 [patent_doc_number] => 20200190092 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2020-06-18 [patent_title] => SUBSTITUTED PYRAZOLO[3,4-d]PYRIMIDINES AS KINASE INHIBITORS [patent_app_type] => utility [patent_app_number] => 16/708340 [patent_app_country] => US [patent_app_date] => 2019-12-09 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 21135 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -16 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16708340 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/708340
Substituted pyrazolo[3,4-d]pyrimidines as kinase inhibitors Dec 8, 2019 Issued
Array ( [id] => 16176879 [patent_doc_number] => 20200223847 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2020-07-16 [patent_title] => SUBSTITUTED-QUINOXALINE-TYPE BRIDGED-PIPERIDINE COMPOUNDS AND THE USES THEREOF [patent_app_type] => utility [patent_app_number] => 16/705814 [patent_app_country] => US [patent_app_date] => 2019-12-06 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 37541 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -9 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16705814 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/705814
Pharmaceutical salts of substituted-quinoxaline-type bridged-piperidine compounds Dec 5, 2019 Issued
Array ( [id] => 17414011 [patent_doc_number] => 20220048915 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-02-17 [patent_title] => Nitrogen-containing Heterocyclic Compound and Composition Thereof, Preparation Method Therefor, and Application Thereof [patent_app_type] => utility [patent_app_number] => 17/295876 [patent_app_country] => US [patent_app_date] => 2019-12-02 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 25283 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -21 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17295876 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/295876
Nitrogen-containing Heterocyclic Compound and Composition Thereof, Preparation Method Therefor, and Application Thereof Dec 1, 2019 Abandoned
Array ( [id] => 16190690 [patent_doc_number] => 20200231539 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2020-07-23 [patent_title] => MULTIPLE CYCLOADDITION REACTIONS FOR LABELING OF MOLECULES [patent_app_type] => utility [patent_app_number] => 16/692604 [patent_app_country] => US [patent_app_date] => 2019-11-22 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 31619 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -11 [patent_words_short_claim] => 52 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16692604 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/692604
MULTIPLE CYCLOADDITION REACTIONS FOR LABELING OF MOLECULES Nov 21, 2019 Abandoned
Array ( [id] => 17335977 [patent_doc_number] => 20220002308 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-01-06 [patent_title] => AROMATIC RING-LINKED DIOXINO-QUINAZOLINE OR DIOXINO-QUINOLINE COMPOUNDS, COMPOSITIONS AND USE THEREOF [patent_app_type] => utility [patent_app_number] => 17/293416 [patent_app_country] => US [patent_app_date] => 2019-11-15 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 40729 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -13 [patent_words_short_claim] => 382 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17293416 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/293416
Substituted aromatic ring-linked dioxinoquinazolines and dioxinoquinolines as kinase inhibitors Nov 14, 2019 Issued
Array ( [id] => 16176892 [patent_doc_number] => 20200223860 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2020-07-16 [patent_title] => THE TOTAL SYNTHESIS OF GLUCOSEPANE AND RELATED CHEMICAL REACTIONS, COMPOUNDS AND COMPOSITIONS AND OBTAINED THEREFROM AND METHODS OF TREATMENT [patent_app_type] => utility [patent_app_number] => 16/685856 [patent_app_country] => US [patent_app_date] => 2019-11-15 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 26442 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -19 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16685856 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/685856
THE TOTAL SYNTHESIS OF GLUCOSEPANE AND RELATED CHEMICAL REACTIONS, COMPOUNDS AND COMPOSITIONS AND OBTAINED THEREFROM AND METHODS OF TREATMENT Nov 14, 2019 Abandoned
Array ( [id] => 15618717 [patent_doc_number] => 20200079763 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2020-03-12 [patent_title] => QUINOXALINE AND PYRIDOPYRAZINE DERIVATIVES AS A PI3KB INHIBITORS [patent_app_type] => utility [patent_app_number] => 16/680605 [patent_app_country] => US [patent_app_date] => 2019-11-12 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 80683 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -4 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16680605 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/680605
(R)-8-(1-((3-fluorophenyl)amino)ethyl)-N-(2-hydroxyethyl)-2-morpholinoquinoxaline-6-carboxamide for inhibiting phosphoinositide-3-kinase activity Nov 11, 2019 Issued
Array ( [id] => 16246041 [patent_doc_number] => 10745381 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2020-08-18 [patent_title] => Substituted isoquinolines and phthalazines as rock kinase inhibitors [patent_app_type] => utility [patent_app_number] => 16/676044 [patent_app_country] => US [patent_app_date] => 2019-11-06 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 22112 [patent_no_of_claims] => 19 [patent_no_of_ind_claims] => 2 [patent_words_short_claim] => 15 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16676044 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/676044
Substituted isoquinolines and phthalazines as rock kinase inhibitors Nov 5, 2019 Issued
Array ( [id] => 15524909 [patent_doc_number] => 20200054760 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2020-02-20 [patent_title] => NOVEL PEPTIDIC LINKERS AND CRYPTOPHYCIN CONJUGATES, THEIR PREPARATION AND THEIR THERAPEUTIC USE [patent_app_type] => utility [patent_app_number] => 16/673367 [patent_app_country] => US [patent_app_date] => 2019-11-04 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 51191 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -21 [patent_words_short_claim] => 978 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16673367 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/673367
Cryptophycin antibody conjugates for the treatment of cancer Nov 3, 2019 Issued
Array ( [id] => 15866083 [patent_doc_number] => 20200140445 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2020-05-07 [patent_title] => PYRAZOLOPYRIMIDINE PDE9 INHIBITORS [patent_app_type] => utility [patent_app_number] => 16/670093 [patent_app_country] => US [patent_app_date] => 2019-10-31 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 27142 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -23 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16670093 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/670093
Substituted pyrazolo[3,4-d]pyrimidines as PDE9 inhibitors Oct 30, 2019 Issued
Array ( [id] => 16727828 [patent_doc_number] => 20210094975 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2021-04-01 [patent_title] => RAPAMYCIN ANALOGS AS MTOR INHIBITORS [patent_app_type] => utility [patent_app_number] => 16/669319 [patent_app_country] => US [patent_app_date] => 2019-10-30 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 66176 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -15 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16669319 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/669319
RAPAMYCIN ANALOGS AS MTOR INHIBITORS Oct 29, 2019 Abandoned
Array ( [id] => 17267489 [patent_doc_number] => 11192900 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2021-12-07 [patent_title] => Substituted 1,6-dihydropyridinones and 1,2-dihydroisoquinolinones as bet inhibitors [patent_app_type] => utility [patent_app_number] => 16/669421 [patent_app_country] => US [patent_app_date] => 2019-10-30 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 4 [patent_figures_cnt] => 5 [patent_no_of_words] => 76694 [patent_no_of_claims] => 25 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 875 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16669421 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/669421
Substituted 1,6-dihydropyridinones and 1,2-dihydroisoquinolinones as bet inhibitors Oct 29, 2019 Issued
Array ( [id] => 19897001 [patent_doc_number] => 12274898 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2025-04-15 [patent_title] => Substituted benzodiazepines as antibody-drug conjugates [patent_app_type] => utility [patent_app_number] => 17/289545 [patent_app_country] => US [patent_app_date] => 2019-10-30 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 4 [patent_figures_cnt] => 7 [patent_no_of_words] => 37856 [patent_no_of_claims] => 19 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 268 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17289545 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/289545
Substituted benzodiazepines as antibody-drug conjugates Oct 29, 2019 Issued
Array ( [id] => 16970403 [patent_doc_number] => 11066363 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2021-07-20 [patent_title] => Substituted 6,11-dihydro-5H-benzo[B]carbazoles as inhibitors of ALK and SRPK [patent_app_type] => utility [patent_app_number] => 16/668484 [patent_app_country] => US [patent_app_date] => 2019-10-30 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 8 [patent_figures_cnt] => 12 [patent_no_of_words] => 30538 [patent_no_of_claims] => 6 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 243 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16668484 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/668484
Substituted 6,11-dihydro-5H-benzo[B]carbazoles as inhibitors of ALK and SRPK Oct 29, 2019 Issued
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