Search

Douglas M. Willis

Examiner (ID: 5249, Phone: (571)270-5757 , Office: P/1624 )

Most Active Art Unit
1624
Art Unit(s)
1624
Total Applications
2485
Issued Applications
1796
Pending Applications
148
Abandoned Applications
577

Applications

Application numberTitle of the applicationFiling DateStatus
Array ( [id] => 16649921 [patent_doc_number] => 10927083 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2021-02-23 [patent_title] => Substituted benzimidazoles as inhibitors of transforming growth factor-b kinase [patent_app_type] => utility [patent_app_number] => 16/273786 [patent_app_country] => US [patent_app_date] => 2019-02-12 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 17 [patent_figures_cnt] => 21 [patent_no_of_words] => 28548 [patent_no_of_claims] => 13 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 178 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16273786 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/273786
Substituted benzimidazoles as inhibitors of transforming growth factor-b kinase Feb 11, 2019 Issued
Array ( [id] => 18044823 [patent_doc_number] => 11518764 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2022-12-06 [patent_title] => Substituted heteroaryls as inhibitors of the BCL6 BTB domain protein-protein interaction [patent_app_type] => utility [patent_app_number] => 16/960924 [patent_app_country] => US [patent_app_date] => 2019-02-06 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 82598 [patent_no_of_claims] => 18 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 641 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16960924 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/960924
Substituted heteroaryls as inhibitors of the BCL6 BTB domain protein-protein interaction Feb 5, 2019 Issued
Array ( [id] => 15023311 [patent_doc_number] => 20190322660 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2019-10-24 [patent_title] => SMYD INHIBITORS [patent_app_type] => utility [patent_app_number] => 16/269338 [patent_app_country] => US [patent_app_date] => 2019-02-06 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 43571 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -17 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16269338 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/269338
SMYD INHIBITORS Feb 5, 2019 Abandoned
Array ( [id] => 16711854 [patent_doc_number] => 20210079001 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2021-03-18 [patent_title] => COMPOUNDS AND METHODS FOR THE MODULATION OF AHR [patent_app_type] => utility [patent_app_number] => 16/967100 [patent_app_country] => US [patent_app_date] => 2019-02-05 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 20126 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -17 [patent_words_short_claim] => 271 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16967100 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/967100
Substituted imidazo[1,5-a]pyrazines and [1,2,4]triazolo[4,3-a]pyrazines for the modulation of AhR Feb 4, 2019 Issued
Array ( [id] => 16854880 [patent_doc_number] => 20210155625 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2021-05-27 [patent_title] => 2,3,4,5-TETRAHYDRO-1H-PYRIDO[4, 3-b]INDOLE INHIBITORS OF cGAS FOR TREATING AUTOINFLAMMATORY DISEASES [patent_app_type] => utility [patent_app_number] => 16/967656 [patent_app_country] => US [patent_app_date] => 2019-02-05 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 17587 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -17 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16967656 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/967656
Substituted pyrido[4,3-b]indoles and azepino[4,5-b]indoles as inhibitors of cGAS Feb 4, 2019 Issued
Array ( [id] => 16613600 [patent_doc_number] => 20210032253 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2021-02-04 [patent_title] => PYRAZOLO[1,5-A][1,3,5]TRIAZINE-2-AMINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF [patent_app_type] => utility [patent_app_number] => 16/967370 [patent_app_country] => US [patent_app_date] => 2019-02-01 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 24887 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -21 [patent_words_short_claim] => 382 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16967370 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/967370
PYRAZOLO[1,5-A][1,3,5]TRIAZINE-2-AMINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF Jan 31, 2019 Abandoned
Array ( [id] => 15540759 [patent_doc_number] => 10570144 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2020-02-25 [patent_title] => Substituted ureas as prostaglandin EP4 receptor antagonists [patent_app_type] => utility [patent_app_number] => 16/263518 [patent_app_country] => US [patent_app_date] => 2019-01-31 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 10745 [patent_no_of_claims] => 22 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 108 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16263518 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/263518
Substituted ureas as prostaglandin EP4 receptor antagonists Jan 30, 2019 Issued
Array ( [id] => 16613599 [patent_doc_number] => 20210032252 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2021-02-04 [patent_title] => PRC2 Inhibitors [patent_app_type] => utility [patent_app_number] => 16/966708 [patent_app_country] => US [patent_app_date] => 2019-01-29 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 55964 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -19 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16966708 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/966708
Substituted imidazo[1,2-c]pyrimidines as PRC2 inhibitors Jan 28, 2019 Issued
Array ( [id] => 18201161 [patent_doc_number] => 11583532 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2023-02-21 [patent_title] => Triazolopyrimidine derivatives for use as ghrelin o-acyl transferase (GOAT) inhibitors [patent_app_type] => utility [patent_app_number] => 16/966493 [patent_app_country] => US [patent_app_date] => 2019-01-28 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 20900 [patent_no_of_claims] => 23 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 708 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16966493 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/966493
Triazolopyrimidine derivatives for use as ghrelin o-acyl transferase (GOAT) inhibitors Jan 27, 2019 Issued
Array ( [id] => 18289891 [patent_doc_number] => 11618753 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2023-04-04 [patent_title] => Aminopyrrolotriazines as kinase inhibitors [patent_app_type] => utility [patent_app_number] => 16/963886 [patent_app_country] => US [patent_app_date] => 2019-01-24 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 171606 [patent_no_of_claims] => 9 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 535 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16963886 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/963886
Aminopyrrolotriazines as kinase inhibitors Jan 23, 2019 Issued
Array ( [id] => 15293451 [patent_doc_number] => 20190389861 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2019-12-26 [patent_title] => TETRACYCLIC BROMODOMAIN INHIBITORS [patent_app_type] => utility [patent_app_number] => 16/254124 [patent_app_country] => US [patent_app_date] => 2019-01-22 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 81212 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => 0 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16254124 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/254124
TETRACYCLIC BROMODOMAIN INHIBITORS Jan 21, 2019 Abandoned
Array ( [id] => 16525199 [patent_doc_number] => 20200399279 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2020-12-24 [patent_title] => SUBSTITUTED PYRAZOLO[3,4-d]PYRIMIDINE COMPOUNDS AS RET KINASE INHIBITORS [patent_app_type] => utility [patent_app_number] => 16/961973 [patent_app_country] => US [patent_app_date] => 2019-01-18 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 92485 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -11 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16961973 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/961973
Substituted pyrazolo[3,4-d]pyrimidines as RET kinase inhibitors Jan 17, 2019 Issued
Array ( [id] => 18216415 [patent_doc_number] => 11591337 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2023-02-28 [patent_title] => Substituted [1,2,4]triazolo[4,3-a]pyrazines as modulators of mGlu5 receptors [patent_app_type] => utility [patent_app_number] => 16/964337 [patent_app_country] => US [patent_app_date] => 2019-01-17 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 17588 [patent_no_of_claims] => 11 [patent_no_of_ind_claims] => 2 [patent_words_short_claim] => 15 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16964337 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/964337
Substituted [1,2,4]triazolo[4,3-a]pyrazines as modulators of mGlu5 receptors Jan 16, 2019 Issued
Array ( [id] => 18369084 [patent_doc_number] => 11649238 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2023-05-16 [patent_title] => Substituted pyrazolo[1,5-a]pyrimidines as PI4K inhibitors [patent_app_type] => utility [patent_app_number] => 16/961704 [patent_app_country] => US [patent_app_date] => 2019-01-15 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 36191 [patent_no_of_claims] => 46 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 424 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16961704 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/961704
Substituted pyrazolo[1,5-a]pyrimidines as PI4K inhibitors Jan 14, 2019 Issued
Array ( [id] => 16336477 [patent_doc_number] => 10787421 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2020-09-29 [patent_title] => Substituted anilines for treatment of animal diseases [patent_app_type] => utility [patent_app_number] => 16/248110 [patent_app_country] => US [patent_app_date] => 2019-01-15 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 8192 [patent_no_of_claims] => 15 [patent_no_of_ind_claims] => 3 [patent_words_short_claim] => 9 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16248110 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/248110
Substituted anilines for treatment of animal diseases Jan 14, 2019 Issued
Array ( [id] => 16525197 [patent_doc_number] => 20200399277 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2020-12-24 [patent_title] => [1,2,4]TRIAZOLO[4,3-A]PYRAZIN-8-ONE DERIVATIVES [patent_app_type] => utility [patent_app_number] => 16/956826 [patent_app_country] => US [patent_app_date] => 2019-01-13 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 7257 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -11 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16956826 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/956826
Substituted [1,2,4]triazolo[4,3-a]pyrazines as phosphodiesterase inhibitors Jan 12, 2019 Issued
Array ( [id] => 15666355 [patent_doc_number] => 10597395 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2020-03-24 [patent_title] => Preparation of certain substituted 1-(4-fluorophenyl)-4-(2,3,6b,9,10,10a-hexahydro-1H-pyrido[3',4':4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-YL)butan-1-ones and pharmaceutically acceptable salts thereof [patent_app_type] => utility [patent_app_number] => 16/244796 [patent_app_country] => US [patent_app_date] => 2019-01-10 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 20085 [patent_no_of_claims] => 19 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 480 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16244796 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/244796
Preparation of certain substituted 1-(4-fluorophenyl)-4-(2,3,6b,9,10,10a-hexahydro-1H-pyrido[3',4':4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-YL)butan-1-ones and pharmaceutically acceptable salts thereof Jan 9, 2019 Issued
Array ( [id] => 14342035 [patent_doc_number] => 20190152990 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2019-05-23 [patent_title] => POLYCYCLIC CARBAMOYLPYRIDONE DERIVATIVE HAVING HIV INTEGRASE INHIBITORY ACTIVITY [patent_app_type] => utility [patent_app_number] => 16/244441 [patent_app_country] => US [patent_app_date] => 2019-01-10 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 40088 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -15 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16244441 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/244441
POLYCYCLIC CARBAMOYLPYRIDONE DERIVATIVE HAVING HIV INTEGRASE INHIBITORY ACTIVITY Jan 9, 2019 Abandoned
Array ( [id] => 16792937 [patent_doc_number] => 20210122754 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2021-04-29 [patent_title] => AN IMPROVED PROCESS FOR THE PREPARATION OF RIBOCICLIB SUCCINATE AND ITS NOVEL CRYSTALLINE FORMS THEREOF [patent_app_type] => utility [patent_app_number] => 16/962934 [patent_app_country] => US [patent_app_date] => 2019-01-10 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 5741 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -13 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16962934 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/962934
Process for the preparation of ribociclib succinate and its novel crystalline forms thereof Jan 9, 2019 Issued
Array ( [id] => 14309499 [patent_doc_number] => 20190144453 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2019-05-16 [patent_title] => NOVEL QUINAZOLINONE DERIVATIVES INHIBITING PI3K AND PHARMACEUTICAL COMPOSITION CONTAINING SAME [patent_app_type] => utility [patent_app_number] => 16/244368 [patent_app_country] => US [patent_app_date] => 2019-01-10 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 7344 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -7 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 16244368 [rel_patent_id] =>[rel_patent_doc_number] =>)
16/244368
Substituted quinazolinones for inhibiting PI3K Jan 9, 2019 Issued
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