Search

Douglas M. Willis

Examiner (ID: 237, Phone: (571)270-5757 , Office: P/1624 )

Most Active Art Unit
1624
Art Unit(s)
1624
Total Applications
2404
Issued Applications
1763
Pending Applications
141
Abandoned Applications
559

Applications

Application numberTitle of the applicationFiling DateStatus
Array ( [id] => 19955305 [patent_doc_number] => 12325711 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2025-06-10 [patent_title] => 3-(ethoxydifluoromethyl)-6-(5-fluoro-6-(2,2,2-trifluoroethoxy)pyridin-3-yl)-[1,2,4]triazolo[4,3-a]pyrazine as an ion channel modulator [patent_app_type] => utility [patent_app_number] => 18/236156 [patent_app_country] => US [patent_app_date] => 2023-08-21 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 9 [patent_figures_cnt] => 18 [patent_no_of_words] => 49171 [patent_no_of_claims] => 32 [patent_no_of_ind_claims] => 2 [patent_words_short_claim] => 36 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18236156 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/236156
3-(ethoxydifluoromethyl)-6-(5-fluoro-6-(2,2,2-trifluoroethoxy)pyridin-3-yl)-[1,2,4]triazolo[4,3-a]pyrazine as an ion channel modulator Aug 20, 2023 Issued
Array ( [id] => 19043558 [patent_doc_number] => 11932642 [patent_country] => US [patent_kind] => B1 [patent_issue_date] => 2024-03-19 [patent_title] => Substituted pyrido[3',4':4,5]pyrrolo[3,2-b][1,6]naphthyridines as CK2 inhibitors [patent_app_type] => utility [patent_app_number] => 18/236021 [patent_app_country] => US [patent_app_date] => 2023-08-21 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 8913 [patent_no_of_claims] => 11 [patent_no_of_ind_claims] => 2 [patent_words_short_claim] => 13 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18236021 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/236021
Substituted pyrido[3',4':4,5]pyrrolo[3,2-b][1,6]naphthyridines as CK2 inhibitors Aug 20, 2023 Issued
Array ( [id] => 19248631 [patent_doc_number] => 20240199618 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-06-20 [patent_title] => NOVEL N-ACYL-[3-SUBSTITUTED]-[8-SUBSTITUTED]-5,6-DIHYDRO-[1,2,4]TRIAZOLO[4,3-a]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR-MEDIATED DISORDERS [patent_app_type] => utility [patent_app_number] => 18/235976 [patent_app_country] => US [patent_app_date] => 2023-08-21 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 22521 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -6 [patent_words_short_claim] => 71 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18235976 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/235976
NOVEL N-ACYL-[3-SUBSTITUTED]-[8-SUBSTITUTED]-5,6-DIHYDRO-[1,2,4]TRIAZOLO[4,3-a]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR-MEDIATED DISORDERS Aug 20, 2023 Abandoned
Array ( [id] => 19111193 [patent_doc_number] => 20240122943 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-04-18 [patent_title] => METHODS AND COMPOSITIONS FOR REDUCING BODY FAT AND ADIPOCYTES [patent_app_type] => utility [patent_app_number] => 18/450253 [patent_app_country] => US [patent_app_date] => 2023-08-15 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 17212 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => 0 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18450253 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/450253
METHODS AND COMPOSITIONS FOR REDUCING BODY FAT AND ADIPOCYTES Aug 14, 2023 Abandoned
Array ( [id] => 19579843 [patent_doc_number] => 12145939 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2024-11-19 [patent_title] => Substituted [1,2,4]triazolo[4,3-a]pyrazines as ion channel modulators [patent_app_type] => utility [patent_app_number] => 18/365695 [patent_app_country] => US [patent_app_date] => 2023-08-04 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 37414 [patent_no_of_claims] => 19 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 120 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18365695 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/365695
Substituted [1,2,4]triazolo[4,3-a]pyrazines as ion channel modulators Aug 3, 2023 Issued
Array ( [id] => 19246914 [patent_doc_number] => 20240197898 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-06-20 [patent_title] => SUBSTITUTED BENZO[5,6][1,4]DIAZEPINO[1,2-a]INDOLES FOR THE TREATMENT OF PROLIFERATIVE DISORDERS [patent_app_type] => utility [patent_app_number] => 18/229476 [patent_app_country] => US [patent_app_date] => 2023-08-02 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 48434 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -19 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18229476 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/229476
SUBSTITUTED BENZO[5,6][1,4]DIAZEPINO[1,2-a]INDOLES FOR THE TREATMENT OF PROLIFERATIVE DISORDERS Aug 1, 2023 Pending
Array ( [id] => 18932262 [patent_doc_number] => 11884668 [patent_country] => US [patent_kind] => B1 [patent_issue_date] => 2024-01-30 [patent_title] => Substituted pyrido[3',4':4,5]pyrrolo[2,3-c]quinolines as CK2 inhibitors [patent_app_type] => utility [patent_app_number] => 18/229399 [patent_app_country] => US [patent_app_date] => 2023-08-02 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 11092 [patent_no_of_claims] => 11 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 432 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18229399 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/229399
Substituted pyrido[3',4':4,5]pyrrolo[2,3-c]quinolines as CK2 inhibitors Aug 1, 2023 Issued
Array ( [id] => 19003581 [patent_doc_number] => 20240067652 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-02-29 [patent_title] => METHOD OF PREPARING INDOLINOBENZODIAZEPINE DERIVATIVES [patent_app_type] => utility [patent_app_number] => 18/229579 [patent_app_country] => US [patent_app_date] => 2023-08-02 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 10393 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -20 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18229579 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/229579
METHOD OF PREPARING INDOLINOBENZODIAZEPINE DERIVATIVES Aug 1, 2023 Abandoned
Array ( [id] => 18922890 [patent_doc_number] => 20240025894 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-01-25 [patent_title] => SUBSTITUTED 5,6,7,8-TETRAHYDROPYRIDO[2,3-D]PYRIMIDINE-2,4-DIONES FOR TREATING CARDIAC DISEASES [patent_app_type] => utility [patent_app_number] => 18/228911 [patent_app_country] => US [patent_app_date] => 2023-08-01 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 29807 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -19 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18228911 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/228911
Substituted 5,6,7,8-tetrahydropyrido[2,3-d]pyrimidine-2,4-diones for treating cardiac diseases Jul 31, 2023 Issued
Array ( [id] => 19504960 [patent_doc_number] => 12116371 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2024-10-15 [patent_title] => Substituted pyridines as irreversible inhibitors of menin-MLL interaction [patent_app_type] => utility [patent_app_number] => 18/228602 [patent_app_country] => US [patent_app_date] => 2023-07-31 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 5 [patent_figures_cnt] => 8 [patent_no_of_words] => 57977 [patent_no_of_claims] => 14 [patent_no_of_ind_claims] => 2 [patent_words_short_claim] => 11 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18228602 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/228602
Substituted pyridines as irreversible inhibitors of menin-MLL interaction Jul 30, 2023 Issued
Array ( [id] => 18964131 [patent_doc_number] => 11897881 [patent_country] => US [patent_kind] => B1 [patent_issue_date] => 2024-02-13 [patent_title] => Substituted pyrido[3,4-b]indole-3-carboxylic acids as CK2 inhibitors [patent_app_type] => utility [patent_app_number] => 18/228609 [patent_app_country] => US [patent_app_date] => 2023-07-31 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 9264 [patent_no_of_claims] => 15 [patent_no_of_ind_claims] => 4 [patent_words_short_claim] => 15 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18228609 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/228609
Substituted pyrido[3,4-b]indole-3-carboxylic acids as CK2 inhibitors Jul 30, 2023 Issued
Array ( [id] => 18752393 [patent_doc_number] => 20230355630 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2023-11-09 [patent_title] => SOLID PHARMACEUTICAL COMPOSITIONS COMPRISING BIOPTERIN DERIVATIVES AND USES OF SUCH COMPOSITIONS [patent_app_type] => utility [patent_app_number] => 18/224515 [patent_app_country] => US [patent_app_date] => 2023-07-20 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 13710 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -16 [patent_words_short_claim] => 199 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18224515 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/224515
Process for preparing solutions comprising biopterin derivatives Jul 19, 2023 Issued
Array ( [id] => 18879024 [patent_doc_number] => 20240002393 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-01-04 [patent_title] => SUBSTITUTED BENZO[f][l ,2,4JTRIAZOL0[4,3-a][l ,4JDIAZEPINES AS GABA A GAMMA! POSITIVE ALLOSTERIC MODULATORS [patent_app_type] => utility [patent_app_number] => 18/355538 [patent_app_country] => US [patent_app_date] => 2023-07-20 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 16472 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -11 [patent_words_short_claim] => 45 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18355538 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/355538
SUBSTITUTED BENZO[f][l ,2,4JTRIAZOL0[4,3-a][l ,4JDIAZEPINES AS GABA A GAMMA! POSITIVE ALLOSTERIC MODULATORS Jul 19, 2023 Pending
Array ( [id] => 18752393 [patent_doc_number] => 20230355630 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2023-11-09 [patent_title] => SOLID PHARMACEUTICAL COMPOSITIONS COMPRISING BIOPTERIN DERIVATIVES AND USES OF SUCH COMPOSITIONS [patent_app_type] => utility [patent_app_number] => 18/224515 [patent_app_country] => US [patent_app_date] => 2023-07-20 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 13710 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -16 [patent_words_short_claim] => 199 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18224515 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/224515
Process for preparing solutions comprising biopterin derivatives Jul 19, 2023 Issued
Array ( [id] => 18871149 [patent_doc_number] => 11858934 [patent_country] => US [patent_kind] => B1 [patent_issue_date] => 2024-01-02 [patent_title] => Substituted pyrido[4',3':5,6]pyrimido[1,2-a]indoles as CK2 inhibitors [patent_app_type] => utility [patent_app_number] => 18/223002 [patent_app_country] => US [patent_app_date] => 2023-07-17 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 8958 [patent_no_of_claims] => 15 [patent_no_of_ind_claims] => 3 [patent_words_short_claim] => 15 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18223002 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/223002
Substituted pyrido[4',3':5,6]pyrimido[1,2-a]indoles as CK2 inhibitors Jul 16, 2023 Issued
Array ( [id] => 18837688 [patent_doc_number] => 11845749 [patent_country] => US [patent_kind] => B1 [patent_issue_date] => 2023-12-19 [patent_title] => Substituted pyrido[4',3':5,6]pyrazino[1,2-a]indoles as anticancer agents [patent_app_type] => utility [patent_app_number] => 18/221438 [patent_app_country] => US [patent_app_date] => 2023-07-13 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 8839 [patent_no_of_claims] => 15 [patent_no_of_ind_claims] => 3 [patent_words_short_claim] => 15 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18221438 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/221438
Substituted pyrido[4',3':5,6]pyrazino[1,2-a]indoles as anticancer agents Jul 12, 2023 Issued
Array ( [id] => 18932261 [patent_doc_number] => 11884667 [patent_country] => US [patent_kind] => B1 [patent_issue_date] => 2024-01-30 [patent_title] => Substituted pyrrolo[2,3-c][2,7]naphthyridines as CK2 inhibitors [patent_app_type] => utility [patent_app_number] => 18/221590 [patent_app_country] => US [patent_app_date] => 2023-07-13 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 10158 [patent_no_of_claims] => 11 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 301 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18221590 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/221590
Substituted pyrrolo[2,3-c][2,7]naphthyridines as CK2 inhibitors Jul 12, 2023 Issued
Array ( [id] => 19097666 [patent_doc_number] => 20240116894 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-04-11 [patent_title] => PROTEASOME ACTIVITY ENHANCING COMPOUNDS [patent_app_type] => utility [patent_app_number] => 18/351264 [patent_app_country] => US [patent_app_date] => 2023-07-12 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 26118 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -18 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18351264 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/351264
PROTEASOME ACTIVITY ENHANCING COMPOUNDS Jul 11, 2023 Abandoned
Array ( [id] => 19248629 [patent_doc_number] => 20240199616 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-06-20 [patent_title] => BICYCLIC COMPOUNDS AS ALLOSTERIC SHP2 INHIBITORS [patent_app_type] => utility [patent_app_number] => 18/220196 [patent_app_country] => US [patent_app_date] => 2023-07-10 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 81040 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -34 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18220196 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/220196
Substituted pyrazolopyrazines, imidazopyrazines and [1,2,4]triazolopyrazines as allosteric SHP2 inhibitors Jul 9, 2023 Issued
Array ( [id] => 20129134 [patent_doc_number] => 12371436 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2025-07-29 [patent_title] => Substituted benzodiazoliums as ENaC inhibitors [patent_app_type] => utility [patent_app_number] => 18/345840 [patent_app_country] => US [patent_app_date] => 2023-06-30 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 7 [patent_figures_cnt] => 13 [patent_no_of_words] => 63090 [patent_no_of_claims] => 24 [patent_no_of_ind_claims] => 3 [patent_words_short_claim] => 1177 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18345840 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/345840
Substituted benzodiazoliums as ENaC inhibitors Jun 29, 2023 Issued
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