Search

J. Casimer Jacyna

Examiner (ID: 1992, Phone: (469)295-9095 , Office: P/3754 )

Most Active Art Unit
3754
Art Unit(s)
3754, 2403, 3751, 2899, 3105
Total Applications
3753
Issued Applications
2853
Pending Applications
166
Abandoned Applications
747

Applications

Application numberTitle of the applicationFiling DateStatus
Array ( [id] => 19083116 [patent_doc_number] => 20240109917 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-04-04 [patent_title] => PYRAZOLOTHIAZOLE CARBOXAMIDES AND THEIR USES AS PDGFR INHIBITORS [patent_app_type] => utility [patent_app_number] => 18/258675 [patent_app_country] => US [patent_app_date] => 2021-12-22 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 156746 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -23 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18258675 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/258675
PYRAZOLOTHIAZOLE CARBOXAMIDES AND THEIR USES AS PDGFR INHIBITORS Dec 21, 2021 Abandoned
Array ( [id] => 17533558 [patent_doc_number] => 20220112167 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-04-14 [patent_title] => Method For Preparing Aryl 2-Tetrazol-1-Yl Keto With Improved Selectivity [patent_app_type] => utility [patent_app_number] => 17/555801 [patent_app_country] => US [patent_app_date] => 2021-12-20 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 4775 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -13 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17555801 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/555801
Method For Preparing Aryl 2-Tetrazol-1-Yl Keto With Improved Selectivity Dec 19, 2021 Abandoned
Array ( [id] => 18987684 [patent_doc_number] => 20240059653 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-02-22 [patent_title] => METHOD OF SYNTHESIZING INDOLE COMPOUNDS [patent_app_type] => utility [patent_app_number] => 18/259578 [patent_app_country] => US [patent_app_date] => 2021-12-17 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 26508 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -83 [patent_words_short_claim] => 19 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18259578 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/259578
Method of synthesizing indole compounds Dec 16, 2021 Issued
Array ( [id] => 18953723 [patent_doc_number] => 20240042050 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-02-08 [patent_title] => ANTI-HER2 IMMUNOCONJUGATES, AND USES THEREOF [patent_app_type] => utility [patent_app_number] => 18/038897 [patent_app_country] => US [patent_app_date] => 2021-12-10 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 21704 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -34 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18038897 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/038897
ANTI-HER2 IMMUNOCONJUGATES, AND USES THEREOF Dec 9, 2021 Pending
Array ( [id] => 18879035 [patent_doc_number] => 20240002404 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-01-04 [patent_title] => SALT OF PYRROLOPYRIMIDINE COMPOUND, CRYSTALLINE FORM THEREOF, AND APPLICATION THEREOF [patent_app_type] => utility [patent_app_number] => 18/254186 [patent_app_country] => US [patent_app_date] => 2021-12-06 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 14721 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -17 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18254186 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/254186
SALT OF PYRROLOPYRIMIDINE COMPOUND, CRYSTALLINE FORM THEREOF, AND APPLICATION THEREOF Dec 5, 2021 Pending
Array ( [id] => 17627212 [patent_doc_number] => 20220162227 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-05-26 [patent_title] => METHODS FOR THE PREPARATION OF 1,3-BENZODIOXOLE HETEROCYCLIC COMPOUNDS [patent_app_type] => utility [patent_app_number] => 17/539715 [patent_app_country] => US [patent_app_date] => 2021-12-01 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 9188 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -19 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17539715 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/539715
Methods for the preparation of 1,3-benzodioxole heterocyclic compounds Nov 30, 2021 Issued
Array ( [id] => 17807319 [patent_doc_number] => 20220259154 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-08-18 [patent_title] => COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF ANDROGEN RECEPTOR [patent_app_type] => utility [patent_app_number] => 17/539679 [patent_app_country] => US [patent_app_date] => 2021-12-01 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 50764 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -4 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17539679 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/539679
Compounds and methods for the targeted degradation of androgen receptor Nov 30, 2021 Issued
Array ( [id] => 17929695 [patent_doc_number] => 20220324820 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-10-13 [patent_title] => METHODS AND COMPOSITIONS FOR GAMMA-GLUTAMYL CYCLE MODULATION [patent_app_type] => utility [patent_app_number] => 17/537266 [patent_app_country] => US [patent_app_date] => 2021-11-29 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 21482 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -24 [patent_words_short_claim] => 20 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17537266 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/537266
METHODS AND COMPOSITIONS FOR GAMMA-GLUTAMYL CYCLE MODULATION Nov 28, 2021 Pending
Array ( [id] => 18853879 [patent_doc_number] => 11851440 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2023-12-26 [patent_title] => Modulators of eukaryotic initiation factor 2B, compositions and methods [patent_app_type] => utility [patent_app_number] => 17/531039 [patent_app_country] => US [patent_app_date] => 2021-11-19 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 55266 [patent_no_of_claims] => 18 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 56 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17531039 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/531039
Modulators of eukaryotic initiation factor 2B, compositions and methods Nov 18, 2021 Issued
Array ( [id] => 18861808 [patent_doc_number] => 20230416243 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2023-12-28 [patent_title] => Process for Preparing Heterocyclic Methanone Compounds and AZA-Bicyclo Intermediates Thereof [patent_app_type] => utility [patent_app_number] => 18/252025 [patent_app_country] => US [patent_app_date] => 2021-11-05 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 17220 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -17 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18252025 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/252025
Process for Preparing Heterocyclic Methanone Compounds and AZA-Bicyclo Intermediates Thereof Nov 4, 2021 Pending
Array ( [id] => 18153041 [patent_doc_number] => 11566001 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2023-01-31 [patent_title] => Hepatitis B capsid assembly modulators [patent_app_type] => utility [patent_app_number] => 17/514578 [patent_app_country] => US [patent_app_date] => 2021-10-29 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 38757 [patent_no_of_claims] => 11 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 100 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17514578 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/514578
Hepatitis B capsid assembly modulators Oct 28, 2021 Issued
Array ( [id] => 19717279 [patent_doc_number] => 12202802 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2025-01-21 [patent_title] => Styryl quinolinium, process for their preparation and use thereof as fluorescent probes for imaging [patent_app_type] => utility [patent_app_number] => 17/507028 [patent_app_country] => US [patent_app_date] => 2021-10-21 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 7 [patent_figures_cnt] => 16 [patent_no_of_words] => 6222 [patent_no_of_claims] => 2 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 7 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17507028 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/507028
Styryl quinolinium, process for their preparation and use thereof as fluorescent probes for imaging Oct 20, 2021 Issued
Array ( [id] => 17385501 [patent_doc_number] => 20220033353 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-02-03 [patent_title] => PROCESS FOR PREPARING CYANOACETATES [patent_app_type] => utility [patent_app_number] => 17/503914 [patent_app_country] => US [patent_app_date] => 2021-10-18 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 1487 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -16 [patent_words_short_claim] => 47 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17503914 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/503914
Process for preparing cyanoacetates Oct 17, 2021 Issued
Array ( [id] => 17385498 [patent_doc_number] => 20220033350 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-02-03 [patent_title] => PROCESS FOR PREPARING CYANOACETATES [patent_app_type] => utility [patent_app_number] => 17/503897 [patent_app_country] => US [patent_app_date] => 2021-10-18 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 1884 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -28 [patent_words_short_claim] => 60 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17503897 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/503897
Process for preparing cyanoacetates Oct 17, 2021 Issued
Array ( [id] => 18986486 [patent_doc_number] => 20240058455 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-02-22 [patent_title] => BIOORTHOGONAL LINKERS AND REACTIONS [patent_app_type] => utility [patent_app_number] => 18/247571 [patent_app_country] => US [patent_app_date] => 2021-10-04 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 46359 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -59 [patent_words_short_claim] => 189 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18247571 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/247571
BIOORTHOGONAL LINKERS AND REACTIONS Oct 3, 2021 Pending
Array ( [id] => 17561618 [patent_doc_number] => 20220125767 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-04-28 [patent_title] => THIAZOLIDE COMPOUNDS FOR TREATING VIRAL INFECTIONS [patent_app_type] => utility [patent_app_number] => 17/491878 [patent_app_country] => US [patent_app_date] => 2021-10-01 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 9977 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -17 [patent_words_short_claim] => 71 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17491878 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/491878
THIAZOLIDE COMPOUNDS FOR TREATING VIRAL INFECTIONS Sep 30, 2021 Abandoned
Array ( [id] => 19343525 [patent_doc_number] => 20240252488 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-08-01 [patent_title] => MLKL BINDING OR DEGRADING COMPOUND AND PHARMACEUTICAL USE THEREOF [patent_app_type] => utility [patent_app_number] => 18/246773 [patent_app_country] => US [patent_app_date] => 2021-09-27 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 88880 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -26 [patent_words_short_claim] => 287 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18246773 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/246773
MLKL BINDING OR DEGRADING COMPOUND AND PHARMACEUTICAL USE THEREOF Sep 26, 2021 Pending
Array ( [id] => 17343620 [patent_doc_number] => 20220009951 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-01-13 [patent_title] => TORSEMIDE PHOSPHATE PRODRUG, PREPARATION METHOD AND COMPOSITION THEREOF [patent_app_type] => utility [patent_app_number] => 17/482827 [patent_app_country] => US [patent_app_date] => 2021-09-23 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 2533 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -8 [patent_words_short_claim] => 13 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17482827 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/482827
TORSEMIDE PHOSPHATE PRODRUG, PREPARATION METHOD AND COMPOSITION THEREOF Sep 22, 2021 Abandoned
Array ( [id] => 19083052 [patent_doc_number] => 20240109853 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2024-04-04 [patent_title] => ALPHA PROTEIN KINASE 1 INHIBITORS AND METHODS OF USE [patent_app_type] => utility [patent_app_number] => 18/246586 [patent_app_country] => US [patent_app_date] => 2021-09-23 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 48511 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -21 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18246586 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/246586
ALPHA PROTEIN KINASE 1 INHIBITORS AND METHODS OF USE Sep 22, 2021 Pending
Array ( [id] => 18752384 [patent_doc_number] => 20230355617 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2023-11-09 [patent_title] => SMALL MOLECULE INHIBITORS OF LEMUR TYROSINE KINASE 3 [patent_app_type] => utility [patent_app_number] => 18/026054 [patent_app_country] => US [patent_app_date] => 2021-09-14 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 16416 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -17 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18026054 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/026054
SMALL MOLECULE INHIBITORS OF LEMUR TYROSINE KINASE 3 Sep 13, 2021 Pending
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