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Michael S. Brooke

Examiner (ID: 8555)

Most Active Art Unit
2853
Art Unit(s)
2853
Total Applications
507
Issued Applications
449
Pending Applications
14
Abandoned Applications
44

Applications

Application numberTitle of the applicationFiling DateStatus
Array ( [id] => 20664785 [patent_doc_number] => 12606547 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2026-04-21 [patent_title] => Preparation method of phenylisoxazoline compound [patent_app_type] => utility [patent_app_number] => 18/003906 [patent_app_country] => US [patent_app_date] => 2021-06-30 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 0 [patent_no_of_claims] => 8 [patent_no_of_ind_claims] => 2 [patent_words_short_claim] => 246 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18003906 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/003906
Preparation method of phenylisoxazoline compound Jun 29, 2021 Issued
Array ( [id] => 17314381 [patent_doc_number] => 20210403429 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2021-12-30 [patent_title] => METHODS OF SYNTHESIZING 2-[4-[(2,3,4-TRIMETHOXYPHENYL)METHYL]PIPERAZIN-1-YL]ETHYL PYRIDINE-3-CARBOXYLATE [patent_app_type] => utility [patent_app_number] => 17/359762 [patent_app_country] => US [patent_app_date] => 2021-06-28 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 6056 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -19 [patent_words_short_claim] => 70 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17359762 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/359762
Methods of synthesizing 2-[4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-1-yl]ethyl pyridine-3-carboxylate Jun 27, 2021 Issued
Array ( [id] => 18148946 [patent_doc_number] => 20230022803 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2023-01-26 [patent_title] => NOVEL CRYSTALLINE FORM OF GPR40 AGONIST [patent_app_type] => utility [patent_app_number] => 17/358319 [patent_app_country] => US [patent_app_date] => 2021-06-25 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 8921 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -10 [patent_words_short_claim] => 39 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17358319 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/358319
NOVEL CRYSTALLINE FORM OF GPR40 AGONIST Jun 24, 2021 Abandoned
Array ( [id] => 18666217 [patent_doc_number] => 11773094 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2023-10-03 [patent_title] => Farnesoid X receptor agonists and uses thereof [patent_app_type] => utility [patent_app_number] => 17/349757 [patent_app_country] => US [patent_app_date] => 2021-06-16 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 60269 [patent_no_of_claims] => 19 [patent_no_of_ind_claims] => 3 [patent_words_short_claim] => 28 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17349757 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/349757
Farnesoid X receptor agonists and uses thereof Jun 15, 2021 Issued
Array ( [id] => 18664227 [patent_doc_number] => 11771089 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2023-10-03 [patent_title] => Large-scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness [patent_app_type] => utility [patent_app_number] => 17/346446 [patent_app_country] => US [patent_app_date] => 2021-06-14 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 28903 [patent_no_of_claims] => 20 [patent_no_of_ind_claims] => 2 [patent_words_short_claim] => 210 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17346446 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/346446
Large-scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness Jun 13, 2021 Issued
Array ( [id] => 19012996 [patent_doc_number] => 11919911 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2024-03-05 [patent_title] => Methyl (r)-2-(fluoromethyl)-5-oxo-4-phenyl-4,5,6,7-tetrahydro-1H-cyclopenta[b]pyridine-3-carboxylate and methyl (r)-2-(fluoromethyl)-5-oxo-4-phenyl-1,4,5,7-tetrahydrofuro[3,4-b]pyridine-3-carboxylate as CAV1.2 activators [patent_app_type] => utility [patent_app_number] => 17/346006 [patent_app_country] => US [patent_app_date] => 2021-06-11 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 9 [patent_figures_cnt] => 9 [patent_no_of_words] => 33746 [patent_no_of_claims] => 22 [patent_no_of_ind_claims] => 4 [patent_words_short_claim] => 7 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17346006 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/346006
Methyl (r)-2-(fluoromethyl)-5-oxo-4-phenyl-4,5,6,7-tetrahydro-1H-cyclopenta[b]pyridine-3-carboxylate and methyl (r)-2-(fluoromethyl)-5-oxo-4-phenyl-1,4,5,7-tetrahydrofuro[3,4-b]pyridine-3-carboxylate as CAV1.2 activators Jun 10, 2021 Issued
Array ( [id] => 18124755 [patent_doc_number] => 20230010367 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2023-01-12 [patent_title] => RELATED SUBSTANCE OF LINAGLIPTIN INTERMEDIATE AND SYNTHESIS METHOD THEREOF [patent_app_type] => utility [patent_app_number] => 17/433618 [patent_app_country] => US [patent_app_date] => 2021-06-09 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 1648 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => 0 [patent_words_short_claim] => 21 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17433618 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/433618
Related substance of linagliptin intermediate and synthesis method thereof Jun 8, 2021 Issued
Array ( [id] => 18511270 [patent_doc_number] => 20230227403 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2023-07-20 [patent_title] => PROCESS FOR SULFONATION OF 2-AMINOETHANOL HYDROGEN SULFATE ESTER TO PRODUCE TAURINE [patent_app_type] => utility [patent_app_number] => 18/000801 [patent_app_country] => US [patent_app_date] => 2021-06-04 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 6352 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -18 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18000801 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/000801
Process for sulfonation of 2-aminoethanol hydrogen sulfate ester to produce taurine Jun 3, 2021 Issued
Array ( [id] => 18478255 [patent_doc_number] => 11691985 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2023-07-04 [patent_title] => Macrocyclic immunomodulators [patent_app_type] => utility [patent_app_number] => 17/338502 [patent_app_country] => US [patent_app_date] => 2021-06-03 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 16898 [patent_no_of_claims] => 20 [patent_no_of_ind_claims] => 2 [patent_words_short_claim] => 757 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17338502 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/338502
Macrocyclic immunomodulators Jun 2, 2021 Issued
Array ( [id] => 18565612 [patent_doc_number] => 20230255939 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2023-08-17 [patent_title] => Antimicrobial Agent for Non-Human Animal [patent_app_type] => utility [patent_app_number] => 18/000424 [patent_app_country] => US [patent_app_date] => 2021-06-02 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 11875 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -18 [patent_words_short_claim] => 339 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 18000424 [rel_patent_id] =>[rel_patent_doc_number] =>)
18/000424
Antimicrobial agent for non-human animal Jun 1, 2021 Issued
Array ( [id] => 18948100 [patent_doc_number] => 11891381 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2024-02-06 [patent_title] => Compounds for the treatment of glycogen storage disorders [patent_app_type] => utility [patent_app_number] => 17/334905 [patent_app_country] => US [patent_app_date] => 2021-05-31 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 91 [patent_figures_cnt] => 58 [patent_no_of_words] => 16438 [patent_no_of_claims] => 10 [patent_no_of_ind_claims] => 3 [patent_words_short_claim] => 23 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17334905 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/334905
Compounds for the treatment of glycogen storage disorders May 30, 2021 Issued
Array ( [id] => 17546615 [patent_doc_number] => 20220117956 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-04-21 [patent_title] => LSD FOR THE TREATMENT OF ALZHEIMER'S DISEASE [patent_app_type] => utility [patent_app_number] => 17/333214 [patent_app_country] => US [patent_app_date] => 2021-05-28 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 8668 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -14 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17333214 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/333214
LSD FOR THE TREATMENT OF ALZHEIMER'S DISEASE May 27, 2021 Abandoned
Array ( [id] => 17292121 [patent_doc_number] => 20210387960 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2021-12-16 [patent_title] => NRF2 ACTIVATOR [patent_app_type] => utility [patent_app_number] => 17/333498 [patent_app_country] => US [patent_app_date] => 2021-05-28 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 31905 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -17 [patent_words_short_claim] => 2 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17333498 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/333498
NRF2 ACTIVATOR May 27, 2021 Abandoned
Array ( [id] => 19076477 [patent_doc_number] => 11945827 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2024-04-02 [patent_title] => Rapafucin derivative compounds and methods of use thereof [patent_app_type] => utility [patent_app_number] => 17/332331 [patent_app_country] => US [patent_app_date] => 2021-05-27 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 63218 [patent_no_of_claims] => 4 [patent_no_of_ind_claims] => 1 [patent_words_short_claim] => 94 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17332331 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/332331
Rapafucin derivative compounds and methods of use thereof May 26, 2021 Issued
Array ( [id] => 20302400 [patent_doc_number] => 12448378 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2025-10-21 [patent_title] => Fluoropyrrolopyridine compound and application thereof [patent_app_type] => utility [patent_app_number] => 17/928295 [patent_app_country] => US [patent_app_date] => 2021-05-26 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 8638 [patent_no_of_claims] => 12 [patent_no_of_ind_claims] => 2 [patent_words_short_claim] => 18 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17928295 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/928295
Fluoropyrrolopyridine compound and application thereof May 25, 2021 Issued
Array ( [id] => 17482072 [patent_doc_number] => 20220089576 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2022-03-24 [patent_title] => ENANTIOMERICALLY PURIFIED GPER AGONIST FOR USE IN TREATING DISEASE STATES AND CONDITIONS [patent_app_type] => utility [patent_app_number] => 17/328590 [patent_app_country] => US [patent_app_date] => 2021-05-24 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 26869 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -8 [patent_words_short_claim] => 120 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17328590 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/328590
ENANTIOMERICALLY PURIFIED GPER AGONIST FOR USE IN TREATING DISEASE STATES AND CONDITIONS May 23, 2021 Abandoned
Array ( [id] => 18664845 [patent_doc_number] => 11771710 [patent_country] => US [patent_kind] => B2 [patent_issue_date] => 2023-10-03 [patent_title] => Method to treat lipid dysregulation by modulation of proprotein convertase subtilisin/kexin type 9 (PCSK9) protein activity with small molecule ligands [patent_app_type] => utility [patent_app_number] => 17/323260 [patent_app_country] => US [patent_app_date] => 2021-05-18 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 4 [patent_figures_cnt] => 4 [patent_no_of_words] => 16530 [patent_no_of_claims] => 13 [patent_no_of_ind_claims] => 3 [patent_words_short_claim] => 38 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => patent [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17323260 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/323260
Method to treat lipid dysregulation by modulation of proprotein convertase subtilisin/kexin type 9 (PCSK9) protein activity with small molecule ligands May 17, 2021 Issued
Array ( [id] => 17227068 [patent_doc_number] => 20210353624 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2021-11-18 [patent_title] => METHOD OF TREATING CANCER WITH TELOTRISAT OR A PRODRUG THEREOF [patent_app_type] => utility [patent_app_number] => 17/317120 [patent_app_country] => US [patent_app_date] => 2021-05-11 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 12674 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -26 [patent_words_short_claim] => 46 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17317120 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/317120
METHOD OF TREATING CANCER WITH TELOTRISAT OR A PRODRUG THEREOF May 10, 2021 Abandoned
Array ( [id] => 17213067 [patent_doc_number] => 20210346403 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2021-11-11 [patent_title] => USE OF COMPOUNDS THAT TARGET MINERALOCORTICOID RECEPTORS FOR TREATING COVID-19 [patent_app_type] => utility [patent_app_number] => 17/314727 [patent_app_country] => US [patent_app_date] => 2021-05-07 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 2798 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -13 [patent_words_short_claim] => 15 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17314727 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/314727
USE OF COMPOUNDS THAT TARGET MINERALOCORTICOID RECEPTORS FOR TREATING COVID-19 May 6, 2021 Abandoned
Array ( [id] => 17035012 [patent_doc_number] => 20210251970 [patent_country] => US [patent_kind] => A1 [patent_issue_date] => 2021-08-19 [patent_title] => COMPOSITIONS AND METHODS FOR STORAGE STABLE OPHTHALMIC DRUGS [patent_app_type] => utility [patent_app_number] => 17/242398 [patent_app_country] => US [patent_app_date] => 2021-04-28 [patent_effective_date] => 0000-00-00 [patent_drawing_sheets_cnt] => 0 [patent_figures_cnt] => 0 [patent_no_of_words] => 26239 [patent_no_of_claims] => 0 [patent_no_of_ind_claims] => -22 [patent_words_short_claim] => 100 [patent_maintenance] => 1 [patent_no_of_assignments] => 0 [patent_current_assignee] =>[type] => publication [pdf_file] =>[firstpage_image] =>[orig_patent_app_number] => 17242398 [rel_patent_id] =>[rel_patent_doc_number] =>)
17/242398
COMPOSITIONS AND METHODS FOR STORAGE STABLE OPHTHALMIC DRUGS Apr 27, 2021 Abandoned
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