Date Field | Doc. No. | Party | Description |
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Jul 29, 2016 | 2404 | | Ex. 2404 Download |
Jul 29, 2016 | 2403 | | Ex. 2403 Download |
Jul 29, 2016 | 2402 | | Ex. 2402 Download |
Jul 29, 2016 | 2401 | | Ex. 2401 Download |
Jun 28, 2016 | 1034 | petitioner | Exhibit 1034 - Transcript of June 17 2016 Conference Call Download |
Jun 7, 2016 | 1033 | petitioner | Exhibit 1033 Transcript of June 1 2016 Conference Call Download |
May 10, 2016 | 1032 | petitioner | U.S. Patent No. 5,258,389 Download |
May 10, 2016 | 1031 | petitioner | Curriculum Vitae of Steven W. Baldwin Download |
May 10, 2016 | 1030 | petitioner | Declaration of Steven W. Baldwin, Ph.D. in Support of Petition for Inter Partes Review of U.S. Patent No. 5,665,772 Download |
May 10, 2016 | 1029 | petitioner | Stephen W. Michnick et al., Solution Structure of FKBP, a Rotamase Enzyme and Receptor for FK506 and Rapamycin, 252 SCI. 836 1991 Download |
May 10, 2016 | 1028 | petitioner | Yoshihiko Nisibata et al., Automatic Creation of Drug Candidate Structures Based on Receptor Structure Starting Point for Artificial Lead Generation 47 TETRAHEDRON 8985 1991 Download |
May 10, 2016 | 1027 | petitioner | Michael L. Connolly, Solvent Accessible Surfaces of Proteins and Nucleic Acids, 221 SCI. 709 1983 Download |
May 10, 2016 | 1026 | petitioner | Julian Tirado Rives and William L Jorgensen Molecular Dynamics of Proteins with the OPLS Potential Functions. Simulation of the Third Domain of Silver Pheasant Ovomucoid in Water, 112 J. AM. CHEMICAL SOCY 2773 1990 Download |
May 10, 2016 | 1025 | petitioner | William L Jorgensen and Julian Tirado Rives The OPLS Potential Functions for Protein. Energy Minimizations for Crystals of Cyclic Peptides and Crambin 110 J. AM. CHEMICAL SOCY 1657 1988 Download |
May 10, 2016 | 1024 | petitioner | Michael G. Rossmann et al., Three-Dimensional Coordinates from Stereodiagrams of Molecular Structures, B36 ACTA CRYSTALLOGRAPHICA 819 1980 Download |
May 10, 2016 | 1023 | petitioner | R. Stern et al., Rigid rod polymers with flexible side chains, 32 POLYMER 2096 1991 Download |
May 10, 2016 | 1022 | petitioner | M Ballauff,Phase Equilibria in Rodlike Systems with Flexible Side Chains 19 MACROMOLECULES 1366 1986 Download |
May 10, 2016 | 1021 | petitioner | Thomas W Bell Construction of a Soluble Heptacyclic Terpyridine 51 J ORGANIC CHEMISTRY 764 1986 Download |
May 10, 2016 | 1020 | petitioner | Michelle L Lamb et al Estimation of Binding Affinities of FKBP12 Inhibitors Using a Linear Response Method 7 BIOORGANIC AND MEDICINAL CHEMISTRY 851 1999 Download |
May 10, 2016 | 1019 | petitioner | Michelle Lamb and William L Jorgensen Investigations of Neurotrophic Inhibitors of FK506 Binding Protein via Monte Carlo Simulations 41 J.MEDCHEMISTRY 3928 1998 Download |
May 10, 2016 | 1018 | petitioner | Modesto Orozco et al Mechanism for the Rotamase Activity of FK506 Binding Protein from Molecular Dynamics Simulations 32 BIOCHEMISTRY 12864 1993 Download |
May 10, 2016 | 1017 | petitioner | William L Jorgensen Rusting of the Lock and Key Model for ProteinLigand Binding 254 SCI 954 1991 Download |
May 10, 2016 | 1016 | petitioner | Julianto Pranata and William L. Jorgensen, Computational Studies on FK506 Conformational Search and Molecular Dynamics Simulation in Water, 113 J. AM. CHEMICAL SOCY 9483 1991 Download |
May 10, 2016 | 1015 | petitioner | Silverman Chapter 2 Drug Discovery Design and Development THE ORGANIC CHEMISTRY OF DRUG DESIGN AND ACTION 4 1992 Download |
May 10, 2016 | 1014 | petitioner | Hans Joachim Böhm LUDI rule based automatic design of new substituents for enzyme inhibitor leads 6 J COMPUTER AIDED MOLECULAR DESIGN 593 1992 Download |
May 10, 2016 | 1013 | petitioner | Joseph B Moon and W Jeffrey Howe Computer Design of Bioactive Molecules A Method for Receptor Based de Novo Ligand Design 11 PROTEINS STRUCTURE FUNCTION AND GENETICS 314 1991 Download |
May 10, 2016 | 1012 | petitioner | Stuart L Schreiber Chemistry and Biology of the Immunophilins and Their Immunosuppressive Ligands 251 SCI 283 1991 Download |
May 10, 2016 | 1011 | petitioner | US Patent No 5100883 Download |
May 10, 2016 | 1010 | petitioner | US Patent No 4650803 Download |
May 10, 2016 | 1009 | petitioner | US Patent No 5233036 Download |
May 10, 2016 | 1008 | petitioner | Thomas L Lemke Chapter 16 Predicting Water Solubility REVIEW OFORGANIC FUNCTIONAL GROUPS 113 2d ed 1988 Download |
May 10, 2016 | 1007 | petitioner | Samuel H Yalkowsky Estimation of Entropies of Fusion of Organic Compounds 18 INDUS AND ENG CHEMISTRY FUNDAMENTALS 1081979 Download |
May 10, 2016 | 1006 | petitioner | Gregory D Van Duyne et al Atomic Structure of the Rapamycin Human Immunophilin FKBP12 Complex 113 J AM CHEMICAL SOC 7433 1991 Download |
May 10, 2016 | 1005 | petitioner | Randall Ellis Morris Rapamycins Antifungal Antitumor Antiproliferative and Immunosuppressive Macrolides 6 TRANSPLANTATION REVIEWS 39 1992 Download |
May 10, 2016 | 1004 | petitioner | Curriculum Vitae of William L Jorgensen Download |
May 10, 2016 | 1003 | petitioner | Declaration of William L. Jorgensen PhD in Support of Petition for Inter Partes Review of US Patent No 5665772 (Part 3 of 5) Download |
May 10, 2016 | 1003 | petitioner | Declaration of William L. Jorgensen PhD in Support of Petition for Inter Partes Review of US Patent No 5665772 (Part 3 of 5) Download |
May 10, 2016 | 1003 | petitioner | Declaration of William L Jorgensen PhD in Support of Petition for Inter Partes Review of US Patent No 5665772 (Part 1 of 5) Download |
May 10, 2016 | 1003 | petitioner | Declaration of William L. Jorgensen PhD in Support of Petition for Inter Partes Review of US Patent No 5665772 (Part 3 of 5) Download |
May 10, 2016 | 1003 | petitioner | Declaration of William L. Jorgensen PhD in Support of Petition for Inter Partes Review of US Patent No 5665772 (Part 3 of 5) Download |
May 10, 2016 | 1003 | petitioner | Declaration of William L. Jorgensen PhD in Support of Petition for Inter Partes Review of US Patent No 5665772 (Part 3 of 5) Download |
May 10, 2016 | 1003 | petitioner | Declaration of William L. Jorgensen PhD in Support of Petition for Inter Partes Review of US Patent No 5665772 (Part 4 of 5) Download |
May 10, 2016 | 1003 | petitioner | Declaration of William L. Jorgensen PhD in Support of Petition for Inter Partes Review of US Patent No 5665772 (Part 2 of 5) Download |
May 10, 2016 | 1003 | petitioner | Declaration of William L. Jorgensen PhD in Support of Petition for Inter Partes Review of US Patent No 5665772 (Part 5 of 5) Download |
May 10, 2016 | 1002 | petitioner | File History for US Patent No. 5665772 (Part 9 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for US Patent No. 5665772 (Part 3 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for US Patent No. 5665772 (Part 9 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for US Patent No. 5665772 (Part 9 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for US Patent No. 5665772 (Part 9 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for US Patent No. 5665772 (Part 9 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for US Patent No. 5665772 (Part 9 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for US Patent No. 5665772 (Part 9 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for US Patent No. 5665772 (Part 9 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for US Patent No. 5665772 (Part 9 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for US Patent No. 5665772 (Part 9 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for US Patent No. 5665772 (Part 6 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for US Patent No. 5665772 (Part 9 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for US Patent No. 5665772 (Part 10 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for US Patent No. 5665772 (Part 5 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for the '772 Patent (Part 12 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for US Patent No. 5665772 (Part 9 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for the '772 Patent (Part 1 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for US Patent No. 5665772 (Part 11 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for the '772 Patent (Part 8 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for the '772 Patent (Part 7 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for US Patent No. 5665772 (Part 13 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for US Patent No. 5665772 (Part 9 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for US Patent No. 5665772 (Part 2 of 13) Download |
May 10, 2016 | 1002 | petitioner | File History for the '772 Patent (Part 4 of 13) Download |
May 10, 2016 | 1001 | petitioner | US Patent No 5665772 Download |
Jan 11, 2018 | 22 | | Final Written Decision (IPR2016-00084) Download |
Oct 27, 2016 | 21 | | Termination Decision Document Download |
Oct 27, 2016 | 20 | | Joined with IPR2016-00084 per Motion (Paper 20) Download |
Oct 27, 2016 | 19 | | Granting, Granting-in-Part, and Denying Motions for Joinder Download |
Jul 29, 2016 | 18 | | Patent Owner's Exhibit List 1 Download |
Jul 29, 2016 | 17 | | Patent Owner's Preliminary Response Download |
Jul 11, 2016 | 16 | | Breckenridge Reply to Opposition to Petitioner Motion for Joinder Download |
Jun 30, 2016 | 15 | board | Order - re Due Date for Preliminary Response Download |
Jun 28, 2016 | 14 | petitioner | Petitioner's Updated Exhibit List Download |
Jun 28, 2016 | 13 | petitioner | Petitioner's Transmittal Letter Accompanying Submission of Exhibit 1034 Download |
Jun 10, 2016 | 12 | patent_own | Patent Owner's Opposition to Breckenridge's Motion For Joinder Download |
Jun 7, 2016 | 11 | petitioner | Petitioner's Updated Exhibit List Download |
Jun 7, 2016 | 10 | petitioner | Petitioner's Transmittal Letter Accompanying Submission of Exhibit 1033 Download |
Jun 3, 2016 | 9 | petitioner | Petitioner's Updated Mandatory Notices Download |
May 31, 2016 | 8 | patent_own | Patent Owner's Mandatory Notices Download |
May 27, 2016 | 7 | potential_ | Power of Attorney Download |
May 13, 2016 | 6 | board | Notice of Filing Date Accorded to Petition Download |
May 10, 2016 | 5 | petitioner | Motion For Joinder Pursuant to 35 USC 315c and 37 CFR 42_122b Download |
May 10, 2016 | 4 | petitioner | Petition For Inter Partes Review of US Patent No 5665772 under 35 USC 311-319 and 37 CFR 42_100 et seq Download |
May 10, 2016 | 3 | petitioner | Expunged Download |
May 10, 2016 | 2 | petitioner | Power of Attorney Download |
May 10, 2016 | 1 | petitioner | Petitioner's Appendix of the Exhibits Download |