Case number IPR2017-01712
Gilead Sciences, Inc. v. Regents of the University of Minnesota > Documents
| Date Field | Doc. No. | Party | Description |
|---|---|---|---|
| Jun 30, 2017 | 1 | Petition for Inter Partes Review of U.S. Patent No. 8,815,830 Download | |
| Jun 30, 2017 | 2 | Petitioner's Power of Attorney Download | |
| Jul 10, 2017 | 3 | Patent Owner's Mandatory Notices Download | |
| Jul 10, 2017 | 4 | Patent Owner's Power of Attorney Download | |
| Jul 29, 2017 | 5 | Notice of Accord Filing Date Download | |
| Sep 11, 2017 | 6 | Petitioner¿¿¿s Motion For Admission Pro Hac Vice Of Nevin M. Gewertz Under 37 C.F.R. ¿¿ 42.10(c) Download | |
| Sep 11, 2017 | 7 | Petitioner's Motion For Admission Pro Hac Vice Of Adam K. Mortara Under 37 C.F.R. 42.10(c) Download | |
| Sep 11, 2017 | 8 | Petitioner's Motion For Admission Pro Hac Vice Of J. Scott McBride Under 37 C.F.R. 42.10(c) Download | |
| Sep 11, 2017 | 9 | Petitioner's Motion For Admission Pro Hac Vice Of Robert S. Schwartz Under 37 C.F.R. 42.10(c) Download | |
| Sep 11, 2017 | 10 | Petitioner's First Amended Exhibit List Download | |
| Sep 12, 2017 | 11 | Petitioner's Submission of Transcript Download | |
| Sep 12, 2017 | 12 | Petitioner's First Amended Mandatory Notices Download | |
| Sep 12, 2017 | 13 | Petitioner's Second Amended Exhibit List Download | |
| Sep 18, 2017 | 14 | Patent Owner's Motion to Dismiss Download | |
| Sep 18, 2017 | 15 | Patent Owner's Corrected Certificate of Service Download | |
| Sep 21, 2017 | 16 | Request for Refund Download | |
| Sep 25, 2017 | 17 | Gilead Sciences, Inc. Opposition to Regents of the University of Minnesota's Motion to Dismiss Download | |
| Sep 28, 2017 | 18 | Patent Owner's Reply in Support of Motion to Dismiss Download | |
| Oct 25, 2017 | 19 | Order - Conduct of the Proceeding - 37 CFR 42.5 Download | |
| Oct 26, 2017 | 20 | Decision Petitioner's Motions for Pro Hac Vice Admission of Nevin M. Gewertz, Adam K. Mortara, J. Scott McBride, and Robert S. Schwartz Download | |
| Nov 8, 2017 | 21 | Patent Owner Notice of Filing Transcript of October 24, 2017 Conference Call Download | |
| Nov 9, 2017 | 22 | Patent Owner's Updated Mandatory Notices Download | |
| Nov 13, 2017 | 23 | Petitioner's Second Amended Mandatory Notices Download | |
| Feb 5, 2018 | 24 | Conduct of the Proceeding Download | |
| Feb 9, 2018 | 25 | Petitioner's Request for Rehearing Download | |
| Feb 9, 2018 | 26 | Petitioner's Third Amended Exhibit List Download | |
| Feb 22, 2018 | 27 | Decision Denying Petitioner's Request for Rehearing Download | |
| May 16, 2018 | 28 | Petitioner's Third Amended Mandatory Notices Download | |
| Dec 5, 2018 | 29 | Petitioner¿¿¿s Fourth Amended Mandatory Notices Download | |
| Aug 21, 2019 | 30 | Decision - 37 C.F.R. 42.71(b) Download | |
| Aug 23, 2019 | 31 | Patent Owner's Notice of Filing Transcript of August 20, 2019 Conference Call Download | |
| Nov 25, 2019 | 32 | Download | |
| Jan 13, 2020 | 33 | Patent Owner's Notice of Denial of Petition for Cert in Regents of the University of Minnesota v. LSI Corp. Download | |
| Jan 14, 2020 | 34 | Denying Patent Owner's Motion to Dismiss Download | |
| Jan 29, 2020 | 35 | Patent Owner's Second Updated Mandatory Notices Download | |
| Jan 29, 2020 | 36 | Patent Owner's Updated Power of Attorney Download | |
| Feb 4, 2020 | 37 | Patent Owner's Unopposed Motion to Substitute Lead Counsel Download | |
| Feb 6, 2020 | 38 | ORDER Granting Patent Owner's Motion to Substitute Lead Counsel Download | |
| Feb 13, 2020 | 39 | Download | |
| Feb 21, 2020 | 40 | Petitioner's Notice Download | |
| Feb 28, 2020 | 41 | Patent Owner's Response to Petitioner's Notice of Ranking Petitions Download | |
| Mar 2, 2020 | 42 | Patent Owner's Preliminary Response Download | |
| Mar 23, 2020 | 43 | Petitioner's Authorized Table of Supplemental Authority Download | |
| Apr 22, 2020 | 44 | Petitioner's Fifth Amended Mandatory Notices Download | |
| Apr 22, 2020 | 45 | Petitioner's Updated Power of Attorney Download | |
| May 28, 2020 | 46 | Decision Granting Institution of Inter Partes Review Download | |
| May 28, 2020 | 47 | Order Conduct of the Proceeding Scheduling Order Download | |
| Jun 24, 2020 | 48 | board | Download |
| Jun 26, 2020 | 49 | patent_own | Joint Notice of Stipulation Modifying Scheduling Order Download |
| Jul 1, 2020 | 50 | patent_own | Patent Owner's Unopposed Motion for Pro Hac Vice Admission of Charles T. Steenburg Download |
| Jul 1, 2020 | 51 | petitioner | Petitioner's Fourth Amended Exhibit List Download |
| Jul 15, 2020 | 52 | patent_own | Notice of Deposition of Dr. Gerardus Josephus Petrus Henricus Boons Download |
| Jul 28, 2020 | 53 | board | Granting Patent Owners Motion for Pro Hac Vice Admission of Charles T. Steenburg 37 C.F.R. sec 42.10 Download |
| Aug 21, 2020 | 54 | patent_own | Patent Owner's Response Download |
| Sep 22, 2020 | 55 | petitioner | Petitioner's Sixth Amended Mandatory Notices Download |
| Sep 22, 2020 | 56 | petitioner | Notice of Deposition of Dr. Andrea Brancale Download |
| Oct 30, 2020 | 57 | petitioner | Petitioner's Reply Download |
| Dec 11, 2020 | 58 | patent_own | Patent Owner's Sur-Reply to Gilead's Reply Download |
| Dec 18, 2020 | 59 | patent_own | Patent Owner's Request for Oral Hearing Download |
| Dec 18, 2020 | 60 | petitioner | Petitioner's Request for Oral Argument Download |
| Jan 7, 2021 | 61 | board | Order - Setting Oral Argument - 37 CFR 42.70 Download |
| Feb 1, 2021 | 62 | patent_own | Patent Owner's Notice of Filing Demonstrative Exhibits Download |
| Feb 1, 2021 | 63 | petitioner | Petitioner's Updated Exhibit List Download |
| Feb 1, 2021 | 64 | petitioner | Petitioner's Objections to Patent Owner's Demonstrative Exhibits Download |
| Feb 2, 2021 | 65 | patent_own | Patent Owner's Objections to Petitioner's Demonstrative Exhibits Download |
| Apr 23, 2021 | 66 | board | Hearing Transcript Download |
| May 21, 2021 | 67 | board | Termination Decision Document Download |
| Jul 23, 2021 | 68 | patent_own | Patent Owner's Notice of Appeal Download |
| Jun 30, 2017 | 1001 | U.S. Patent No. 8,815,830 Download | |
| Jun 30, 2017 | 1002 | File History of U.S. Patent Application No. 14/229,292 Download | |
| Jun 30, 2017 | 1003 | Complaint, Regents of the University of Minnesota v. Gilead Sciences, Inc., Civil Action No. 0:16-cv-02915-SRN-HB (D. Minn., Aug. 29, 2016) Download | |
| Jun 30, 2017 | 1004 | U.S. Patent Application Publication No. 2010/0016251 (Sofia) Download | |
| Jun 30, 2017 | 1005 | U.S. Patent Application No. 13/753,252 Download | |
| Jun 30, 2017 | 1006 | Preliminary Amendment, U.S. Patent Application No. 11/721,325 (Jun. 8, 2007) Download | |
| Jun 30, 2017 | 1007 | International Application No. PCT/US2005/044442 Download | |
| Jun 30, 2017 | 1008 | U.S. Provisional Application No. 60/634,677 Download | |
| Jun 30, 2017 | 1009 | U.S. Patent No. 8,765,935 Download | |
| Jun 30, 2017 | 1010 | U.S. Patent No. 8,399,428 Download | |
| Jun 30, 2017 | 1011 | Declaration of Victor E. Marquez, Ph.D. Download | |
| Jun 30, 2017 | 1012 | Curriculum Vitae of Victor E. Marquez, Ph.D. Download | |
| Jun 30, 2017 | 1013 | Anastasi et al., Current Medicinal Chemistry 2003, 10: 1825-1843 Download | |
| Jun 30, 2017 | 1014 | Calogeropoulou et al., Current Topics in Medicinal Chemistry 2003, 3: 1467-1495 Download | |
| Jun 30, 2017 | 1015 | Cahard et al., Mini-Reviews in Medicinal Chemistry 2004, 4: 371-381 Download | |
| Jun 30, 2017 | 1016 | Highleyman, "Lodenosine trials stopped due to safety concerns," BETA 12(4): 4 (1999) Download | |
| Jun 30, 2017 | 1017 | Sicardi et al., European Journal of Pharmaceutical Sciences, 22: 25-31 (2004) Download | |
| Jun 30, 2017 | 1018 | Kim et al., Molecular Pharmaceutics, 1: 102-111 (2004) Download | |
| Jun 30, 2017 | 1019 | CenterWatch 2005 FDA Approved Drugs Download | |
| Jun 30, 2017 | 1020 | Yoo et al., J. Med. Chem. 2008, 51: 7593-7601 Download | |
| Jun 30, 2017 | 1021 | Pauling, J. Amer. Chem. Soc., 54: 3570-3582 (1932) Download | |
| Sep 11, 2017 | 1022 | Declaration of Nevin M. Gewertz Download | |
| Sep 11, 2017 | 1023 | Declaration of Adam K. Mortara Download | |
| Sep 11, 2017 | 1024 | Declaration of J. Scott McBride Download | |
| Sep 11, 2017 | 1025 | Declaration of Robert S. Schwartz Download | |
| Sep 12, 2017 | 1026 | Transcript of Sept. 11, 2017 Conference Call Download | |
| Feb 9, 2018 | 1027 | Preliminary Amendment, U.S. Patent Application No. 14/229,292, (Mar. 31, 2014) Download | |
| Feb 9, 2018 | 1028 | Order, Regents of the University of Minnesota v. Gilead Sciences, Inc., Civil Action No. 0:16-cv-02915-SRN-HB, D.I. 139 (D. Minn. Jun. 9, 2017) Download | |
| Feb 9, 2018 | 1029 | Stipulated Case Management Statement, Regents of the University of Minnesota v. Gilead Sciences, Inc., 17-cv-6056-VC, D.I. 275 (N.D. Cal. Jan. 2, 2018) Download | |
| Feb 9, 2018 | 1030 | January 26 Email from Counsel for Patent Owner to Board and Counsel for Petitioner Download | |
| Feb 9, 2018 | 1031 | January 26, 2018 Email Chain Between Counsel for Petitioner and Counsel for Patent Owner Download | |
| Feb 9, 2018 | 1032 | January 28, 2018 Email from Counsel for Petitioner to Board and Counsel for Patent Owner Download | |
| Feb 9, 2018 | 1033 | Stipulation and Proposed Order to Exclude Filings From IPR Proceedings, Regents of the Univ. of Calif. v. St. Jude Medical, LLC (N.D. Cal. Feb. 2, 2018) Download | |
| Feb 9, 2018 | 1034 | Order, Regents of the University of Minnesota v. AT&T Mobility LLC (D. Minn. May 19, 2017) Download | |
| Feb 9, 2018 | 1035 | Gilead's Motion to Stay Pending Inter Partes Review, Regents of the University of Minnesota v. Gilead Sciences, Inc., 17-cv-6056-VC, D.I. 297 (N.D. Cal. Feb. 7, 2018) Download | |
| Jul 1, 2020 | 1036 | petitioner | Declaration of Dr. Gerardus Josephus Petrus Henricus Boons Download |
| Oct 30, 2020 | 1037 | petitioner | World Intellectual Property Organization (WIPO) FAQs: Amendments to the PCT Regulations (April 1, 2007) Download |
| Oct 30, 2020 | 1038 | petitioner | Transcript of the October 8, 2020 Deposition of Dr. Andrea Brancale Download |
| Oct 30, 2020 | 1039 | petitioner | Second Declaration of Dr. Gerardus Josephus Petrus Henricus Boons Download |
| Oct 30, 2020 | 1040 | petitioner | Judith Howard et al., How Good is Fluorine as a Hydrogen Bond Acceptor?, Tetrahedron 52(38):12613-22 (1996) Download |
| Oct 30, 2020 | 1041 | petitioner | Florante A. Quiocho, Protein-carbohydrate interactions: basic molecular features, Pure & Appl. Chem. 61(7):1293-1306 (1989) Download |
| Feb 1, 2021 | 1042 | petitioner | Petitioner's Demonstrative Exhibits Download |
| Sep 18, 2017 | 2001 | University of Minnesota Charter Download | |
| Sep 18, 2017 | 2002 | University of Minnesota¿¿¿s Consolidated Financial Statements (2015 & 2016) Download | |
| Sep 18, 2017 | 2003 | Gilead Sciences, Inc.¿¿¿s Answer to Plaintiff¿¿¿s Complaint for Patent Infringement Download | |
| Sep 18, 2017 | 2004 | Patent Assignment Download | |
| Nov 8, 2017 | 2005 | Transcript of October 24, 2017 Conference Call Download | |
| Aug 23, 2019 | 2006 | Transcript of August 20, 2019 Conference Call Download | |
| Jul 1, 2020 | 2007 | patent_own | Declaration of Charles T. Steenburg in Support of Motion for Admission Pro Hac Vice Download |
| Aug 21, 2020 | 2008 | patent_own | Abraham et al., Synthesis and Biological Activity of Aromatic Amino Acid Phosphoramidates of 5-Fluoro-2'-Deoxyuridine and 1-Beta-Arabinofuranosylcytosine: Evidence of Phosphoramidase Activity, 39(23) J. MED. CHEM. 4569-75 (1996) ("Abraham 1996") Download |
| Aug 21, 2020 | 2009 | patent_own | Balzarini et al., Antiretrovirus Specificity and Intracellular Metabolism of 2',3'-Didehydro-2',3'-Dideoxythymidine (Stavudine) and Its 5'-Monophosphate Triester Prodrug So324, 50(5) MOLECULAR PHARMACOLOGY 1207-13 (1996) ("Balzarini 1996") Download |
| Aug 21, 2020 | 2010 | patent_own | Marquez et al., HIV-1 Reverse Transcriptase Can Discriminate between Two Conformationally Locked Carbocyclic AZT Triphosphate Analogues, 120 J. AM. CHEM. SOC. 2780-89 (1998) ("Marquez 1998") Download |
| Aug 21, 2020 | 2011 | patent_own | Lima et al., Structure-Based Analysis of Catalysis and Substrate Definition in the HIT Protein Family, 278(5336) SCIENCE 286-90 (1997) ("Lima 1997") Download |
| Aug 21, 2020 | 2012 | patent_own | Brenner et al., Crystal structures of HINT demonstrate that histidine triad proteins are GalT-related nucleotide-binding proteins, 4(3) NATURE STRUCTURAL BIOLOGY 231-38 (1997) ("Brenner 1997") Download |
| Aug 21, 2020 | 2013 | patent_own | Chang et al., Amino Acid Phosphoramidate Monoesters of 3'-Azido-3'-Deoxythymidine: Relationship Between Antiviral Potency and Intracellular Metabolism, 44(2) J. MED. CHEM. 223-31 (2001) ("Chang 2001") Download |
| Aug 21, 2020 | 2014 | patent_own | Carroll et al., Inhibition of Hepatitis C Virus RNA Replication by 2'- Modified Nucleoside Analogs, 278(14) J. BIO. CHEM. 11979-84 (2003) ("Carroll 2003") Download |
| Aug 21, 2020 | 2015 | patent_own | Marquez et al., Experimental and Structural Evidence that Herpes 1 Kinase and Cellular DNA Polymerase(s) Discriminate on the Basis of Sugar Pucker, 126(2) J. AM. CHEM. SOC. 543-49 (2004) ("Marquez 2004") Download |
| Aug 21, 2020 | 2016 | patent_own | Eldrup et al., Structure-Activity Relationship of Purine Ribonucleosides for Inhibition of Hepatitis C Virus RNA-Dependent RNA Polymerase, 47(9) J. MED. CHEM. 2283-95 (2004) ("Eldrup 2004") Download |
| Aug 21, 2020 | 2017 | patent_own | Kim et al., Monitoring the Intracellular Metabolism of Nucleoside Phosphoramidate Pronucleotides by 31P NMR, 23(1-2) NUCLEOSIDES NUCLEOTIDES NUCLEIC ACIDS 483-93 (2004) ("Kim 2004") Download |
| Aug 21, 2020 | 2018 | patent_own | De Clercq, Antivirals and Antiviral Strategies, 2(9) NATURE REVIEWS MICROBIOLOGY 2(9):704-20 (2004) ("De Clercq 2004") Download |
| Aug 21, 2020 | 2019 | patent_own | De Clercq, Antivirals and Antiviral Strategies (Supplementary Information), 2(9) NATURE REVIEWS MICROBIOLOGY 704-20 (2004) ("De Clercq 2004 Supplemental Information") Download |
| Aug 21, 2020 | 2020 | patent_own | U.S. Patent Publication No. 2005/0009737 ("Clark") Download |
| Aug 21, 2020 | 2021 | patent_own | Clark et al., Design, Synthesis, and Antiviral Activity of 2'-Deoxy-2'-Fluoro-2'-C-Methylcytidine, a Potent Inhibitor of Hepatitis C Virus Replication, 48(14) J. MED. CHEM. 5504-08 (2005) ("Clark 2005") Download |
| Aug 21, 2020 | 2022 | patent_own | Chou et al., 31P NMR and Genetic Analysis Establish hinT as the Only Escherchia coli Purine Nucleoside Phosphoramidase and as Essential for Growth under High Salt Conditions, 280(15) J. BIO. CHEM. 15356-61 (2005) ("Chou 2005") Download |
| Aug 21, 2020 | 2023 | patent_own | Perrone et al., First Example of Phosphoramidate Approach Applied to a 4'-Substituted Purine Nucleoside (4'-Azidoadenosine) 50(22) J. MED. CHEM. 5463-5470 (2007) ("Perrone 2007") Download |
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| Aug 21, 2020 | 2052 | patent_own | Drontle et al., Designing a Pronucleotide Strategem: Lessons from Amino Acid Phosphoramidates of Anticancer and Antiviral Pyrimidines, 4(4) MINI-REVS. IN MED. CHEM. 409-19 (2004) ("Drontle 2004") Download |
| Aug 21, 2020 | 2053 | patent_own | Chou et al., Evidence that Human Histidine Triad Nucleotide Binding Protein 3 (Hint3) Is a Distinct Branch of the Histidine Triad (HIT) Superfamily, 373(4) J. MOLECULAR BIO. 978-89 (2007) ("Chou 2007, Hint3") Download |
| Aug 21, 2020 | 2054 | patent_own | Chou et al., Phosphoramidate Pronucleotides, MOLECULAR PHARMS. 208-17 (2007) ("Chou 2007, Phosphoramidate Pronucleotides") Download |
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| Aug 21, 2020 | 2056 | patent_own | International Publication No. WO 2006/063149 Download |
| Aug 21, 2020 | 2057 | patent_own | Petition for Inter Partes Review, IPR2018-00119 (Filed October 25, 2017) Download |
| Aug 21, 2020 | 2058 | patent_own | Declaration of Dr. Andrea Brancale ("Brancale") Download |
| Aug 21, 2020 | 2059 | patent_own | Curriculum Vitae of Dr. Andrea Brancale Download |
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| Feb 1, 2021 | 2119 | patent_own | Patent Owner's Demonstrative Exhibits Download |
| Aug 21, 2019 | 3001 | Exhibit 3001 Download | |
| Aug 21, 2019 | 3002 | Exhibit 3002 Download | |
| Jun 24, 2020 | 3003 | board | Ex.3003 Download |
