Date Field | Doc. No. | Party | Description |
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Jan 11, 2018 | 22 | | EXPUNGED Download |
Jan 11, 2018 | 21 | | Final Written Decision (IPR2016-00084) Download |
Jan 11, 2018 | 23 | | Decision - Dismissing Requests for Rehearing Download |
Jan 11, 2017 | 20 | | Petitioners' Updated Mandatory Notice Download |
Dec 27, 2016 | 19 | | Petitioner's Request for Rehearing of the Board's Decision Denying Joinder Download |
Dec 9, 2016 | 18 | | Patent Owner's Response To Petitioners' Requests For Reconsideration Download |
Oct 27, 2016 | 16 | | Granting, Granting-in-Part, and Denying Motions for Joinder Download |
Oct 27, 2016 | 17 | | Joined with IPR2016-00084 per Motion (Paper 17) Download |
Jul 29, 2016 | 15 | | Patent Owner's Exhibit List 1 Download |
Jul 29, 2016 | 14 | | Patent Owner's Preliminary Response Download |
Jul 29, 2016 | 2402 | | Ex. 2402 Download |
Jul 29, 2016 | 2403 | | Ex. 2403 Download |
Jul 29, 2016 | 2404 | | Ex. 2404 Download |
Jul 29, 2016 | 2401 | | Ex. 2401 Download |
Jul 27, 2016 | 13 | | Petitioner's Reply in Support of its Motion for Joinder Download |
Jun 30, 2016 | 12 | board | Order - re Due Date for Preliminary Response Download |
Jun 27, 2016 | 11 | patent_own | Patent Owner's Opposition To Motion For Joinder Download |
Jun 23, 2016 | 1032 | petitioner | Transcript of June 17, 2016 Conference Call Download |
Jun 23, 2016 | 9 | petitioner | Petitioner's Transmittal Letter Accompanying Submission of Exhibit 1032 Download |
Jun 23, 2016 | 10 | petitioner | Petitioner's Second Amended Exhibit List Download |
Jun 16, 2016 | 8 | patent_own | Patent Owner's Mandatory Notices Download |
Jun 15, 2016 | 7 | potential_ | Power of Attorney Download |
Jun 8, 2016 | 5 | petitioner | Petitioner's Transmittal Letter Accompanying Submission of Exhibit 1031 Download |
Jun 8, 2016 | 1031 | petitioner | Transcript of June 1, 2016 Conference Call Download |
Jun 8, 2016 | 6 | petitioner | Petitioner's Amended Exhibit List Download |
Jun 6, 2016 | 4 | board | Notice Of Filing Date Accorded To Petition Download |
May 26, 2016 | 1020 | petitioner | Michelle L. Lamb et al., Estimation of Binding Affinities of FKBP12 Inhibitors Using a Linear Response Method, 7 BIOORGANIC and MEDICINAL CHEMISTRY 851 (1999) Download |
May 26, 2016 | 1002 | petitioner | File History for the 772 Patent Download |
May 26, 2016 | 1028 | petitioner | Yoshihiko Nisibata et al., Automatic Creation of Drug Candidate Structures Based on Receptor Structure. Starting Point for Artificial Lead Generation., 47 TETRAHEDRON 8985 (1991) Download |
May 26, 2016 | 1021 | petitioner | Thomas W. Bell, Construction of a Soluble Heptacyclic Terpyridine, 51 J. ORGANIC CHEMISTRY 764 (1986) (Bell) Download |
May 26, 2016 | 1025 | petitioner | William L. Jorgensen and Julian Tirado-Rives, The OPLS Potential Functions for Proteins. Energy Minimizations for Crystals of Cyclic Peptides and Crambin, 110 J. AM. CHEMICAL SOCY 1657 (1988) Download |
May 26, 2016 | 1007 | petitioner | Samuel H. Yalkowsky, Estimation of Entropies of Fusion of Organic Compounds, 18 INDUS. and ENGG CHEMISTRY FUNDAMENTALS 108 (1979) (Yalkowsky) Download |
May 26, 2016 | 1010 | petitioner | U.S. Patent No. 4,650,803 (Stella) Download |
May 26, 2016 | 1009 | petitioner | U.S. Patent No. 5,233,036 (Hughes) Download |
May 26, 2016 | 1004 | petitioner | Curriculum Vitae of William L. Jorgensen Download |
May 26, 2016 | 1006 | petitioner | Gregory D. Van Duyne et al., Atomic Structure of the Rapamycin Human Immunophilin FKBP-12 Complex, 113 J. AM. CHEMICAL SOCY 7433 (1991) (Van Duyne) Download |
May 26, 2016 | 1029 | petitioner | Stephen W. Michnick et al., Solution Structure of FKBP, a Rotamase Enzyme and Receptor for FK506 and Rapamycin, 252 SCI. 836 (1991) Download |
May 26, 2016 | 1027 | petitioner | Michael L. Connolly, Solvent-Accessible Surfaces of Proteins and Nucleic Acids, 221 SCI. 709 (1983) Download |
May 26, 2016 | 1001 | petitioner | U.S. Patent No. 5,665,772 (the 772 Patent) Download |
May 26, 2016 | 1012 | petitioner | Stuart L. Schreiber, Chemistry and Biology of the Immunophilins and Their Immunosuppressive Ligands, 251 SCI. 283 (1991) (Schreiber) Download |
May 26, 2016 | 3 | petitioner | Motion for Joinder Pursuant to 35 USC 315(c) and 37 CFR 42.122(b) Download |
May 26, 2016 | 1024 | petitioner | Michael G. Rossmann et al., Three-Dimensional Coordinates from Stereodiagrams of Molecular Structures, B36 ACTA CRYSTALLOGRAPHICA 819 (1980) (Rossmann) Download |
May 26, 2016 | 1011 | petitioner | U.S. Patent No. 5,100,883 (Schiehser) Download |
May 26, 2016 | 1005 | petitioner | Randall Ellis Morris, Rapamycins - Antifungal, Antitumor, Antiproliferative, and Immunosuppressive Macrolides, 6 TRANSPLANTATION REVIEWS 39 (1992) (Morris) Download |
May 26, 2016 | 1014 | petitioner | Hans-Joachim Böhm, LUDI- rule-based automatic design of newsubstituents for enzyme inhibitor leads, 6 J. COMPUTER-AIDED MOLECULAR DESIGN 593 (1992) (Böhm) Download |
May 26, 2016 | 1016 | petitioner | Julianto Pranata and William L. Jorgensen, Computational Studies on FK506 Conformational Search and Molecular Dynamics Simulation in Water, 113 J. AM. CHEMICAL SOCY 9483 (1991) Download |
May 26, 2016 | 1 | petitioner | Power of Attorney Download |
May 26, 2016 | 1019 | petitioner | Michelle L. Lamb and William L. Jorgensen, Investigations of Neurotrophic Inhibitors of FK506 Binding Protein via Monte Carlo Simulations, 41 J. MED. CHEMISTRY 3928 (1998) Download |
May 26, 2016 | 1013 | petitioner | Joseph B. Moon and W. Jeffrey Howe, Computer Design of Bioactive Molecules - A Method for Receptor-Based de Novo Ligand Design, 11 PROTEINS - STRUCTURE, FUNCTION, and GENETICS 314 (1991) (Moon) Download |
May 26, 2016 | 1026 | petitioner | Julian Tirado-Rives and William L. Jorgensen, Molecular Dynamics of Proteins with the OPLS Potential Functions. Simulation of the Third Domain of Silver Pheasant Ovomucoid in Water, 112 J. AM. CHEMICAL SOCY 2773 (1990) Download |
May 26, 2016 | 1023 | petitioner | R. Stern et al., Rigid rod polymers with flexible side chains, 32 POLYMER 2096 (1991) (Stern) Download |
May 26, 2016 | 1003 | petitioner | Declaration of William L. Jorgensen, Ph.D. in Support of Petition for Inter Partes Review of U.S. Patent No. 5,665,772 Download |
May 26, 2016 | 1017 | petitioner | William L. Jorgensen, Rusting of the Lock and Key Model for Protein-Ligand Binding, 254 SCI. 954 (1991) Download |
May 26, 2016 | 1008 | petitioner | Thomas L. Lemke, Chapter 16 - Predicting Water Solubility, REVIEW OF ORGANIC FUNCTIONAL GROUPS 113 (2d ed. 1988) Download |
May 26, 2016 | 1030 | petitioner | Certificate of Correction for U.S. Patent No. 5,665,772 Download |
May 26, 2016 | 1022 | petitioner | M. Ballauff, Phase Equilibria in Rodlike Systems with Flexible Side Chains, 19 MACROMOLECULES 1366 (1986) (Ballauff) Download |
May 26, 2016 | 1015 | petitioner | Silverman, Chapter 2- Drug Discovery, Design, and Development, THE ORGANIC CHEMISTRY OF DRUG DESIGN and ACTION 4 (1992) (Silverman) Download |
May 26, 2016 | 2 | petitioner | Petition for Inter Partes Review of U.S. Patent No. 5,665,772 Under 35 U.S.C. 311-319 and 37 C.F.R. 42.100 et seq. Download |
May 26, 2016 | 1018 | petitioner | Modesto Orozco et al., Mechanism for the Rotamase Activity of FK506 Binding Protein from Molecular Dynamics Simulations, 32 BIOCHEMISTRY 12864 (1993) Download |